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1-(azepan-1-yl)-3-[(pyrimidin-4-yl)amino]propan-2-ol
8-(2-amino-9H-purin-6-yl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(3aR,6aR)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-methoxy-4-[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-3-carbonitrile
7-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N3-(2,3-dihydro-1H-inden-2-yl)-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
(4aS,7aR)-N,N-diethyl-6,6-dioxo-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
8-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-{2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}acetamide
6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
1,9-dimethyl-4-(4-phenoxybutyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(1S,6R)-9-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-methyl-N-phenyl-4-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}aniline
5-(2-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
2-methoxy-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyridine
2-[3-(5-methylfuran-2-yl)-5-[pyridin-3-yl(pyrrolidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[4-(3-methylphenyl)phenyl]piperidin-4-amine
3-[(2R,3R,6R)-5-(1H-imidazol-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}propanamide
N-methyl-3-[methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})amino]propanamide
2-(1-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-imidazol-2-yl)pyridine
1-(2-methoxyphenyl)-4-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
methyl[(3-methylpyridin-4-yl)methyl]{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-(1H-imidazol-2-yl)piperidine
1-(2-methoxyethyl)-6-methyl-3-({[2-(1H-1,2,4-triazol-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(4-fluoro-1H-indol-1-yl)acetamide
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxamide
N-cyclopentyl-1-(2-methylpropyl)-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(diethylamino)-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
N,N-dimethyl-2-{2-[({1-oxaspiro[4.5]decan-3-yl}carbamoyl)amino]phenyl}acetamide
1-[(4-ethylphenyl)methyl]-5-(1-methyl-1H-pyrazol-3-yl)-1H-1,2,4-triazole
5-{[(3S)-3-ethylmorpholin-4-yl]methyl}-N,N-dimethylpyridin-2-amine
2-{1-[3-(3,4-difluorophenyl)propanoyl]-1,4-diazepan-6-yl}acetic acid
N-cyclopropyl-5-oxo-1-(pyridin-2-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxamide
(3R)-1-(5-ethylthiophene-2-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
8-chloro-2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]quinoline
2-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
[(2S,4R)-4-(dimethylamino)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]methanol
6-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
N-(2-fluoroethyl)-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxypropan-1-one
5-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
5-{4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
dimethyl(3-{2-[1-(pyrrolidine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
3-(dimethylamino)-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]benzamide
N-{[1-(methoxymethyl)cyclopropyl]methyl}-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine