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N-[2-(2-fluorophenyl)ethyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
2-[(3-chlorophenyl)methyl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1,3-benzoxazole-6-carboxamide
2-{5-[1-(methylsulfanyl)ethyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
(4aS,8aR)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-(2-methylpropyl)piperidin-4-amine
2-{1-[(2-ethoxyphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{1-[(2-ethoxyphenyl)methyl]-4-[(8-methoxyquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2,6-dimethylquinoline-4-carboxamide
1-[(2-chlorophenyl)methyl]-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1H-1,2,3-triazole-4-carboxamide
[(1-cyclohexylpiperidin-3-yl)methyl]({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})(pyridin-3-ylmethyl)amine
3-(azepane-1-carbonyl)-N-benzyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(butan-2-yl)-5-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
5-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-4-propylpyrimidine
N-{[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
1-[3-oxo-3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propyl]pyrrolidin-2-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2-methoxyphenyl)acetamide
7-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
[(5-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}thiophen-3-yl)methyl]dimethylamine
[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl](methyl){[2-(trifluoromethyl)phenyl]methyl}amine
1-[(4-tert-butylphenyl)methyl]-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
1-(3,4-dichlorophenyl)-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperazine
methyl 5-[(butan-2-yl)amino]-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(3,5-dimethyl-1-benzofuran-2-yl)-1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazole
3-fluoro-2-methoxy-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)benzamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2-methoxyphenyl)methyl]-N-methylpyrimidin-2-amine
2,6-difluoro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-methoxybenzamide
N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-3-(4-methylphenyl)-3-phenylpropanamide
1-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-2,2-dimethylpropan-1-one
N4-methyl-N4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-(3-phenylpiperidin-1-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}acetamide
6-(3-benzoylpiperidine-1-carbonyl)-2-methyl-1,3-benzothiazole
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
(2S)-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(1R,5R)-6-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
4-{2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1λ6-thiomorpholine-1,1-dione
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(oxan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
[(2-methoxyphenyl)methyl](propyl)(quinoxalin-2-ylmethyl)amine
2-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
N-[2-(2-methoxyethoxy)phenyl]-2-methyl-5-oxo-1,4-diazepane-1-carboxamide
5-cyclopropanecarbonyl-1'-(2-phenylethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
7-(5-chloropyridin-2-yl)-4-[(1-ethylpyrrolidin-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-acetyl-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}piperidine-4-carboxamide
1-ethyl-3-[(4-methoxyphenyl)methyl]-5-[5-(pyrrolidin-1-ylmethyl)furan-2-yl]-1H-1,2,4-triazole
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-methyl-N-(propan-2-yl)-1,3-thiazole-4-carboxamide
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-4-methylpiperazine
N-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide