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N-(2-acetyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-(4-methylphenyl)propanamide
2-cyclopropyl-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl})(quinolin-4-ylmethyl)amine
N-{[4-(dimethylamino)oxan-4-yl]methyl}-1-(furan-2-ylmethyl)piperidine-4-carboxamide
2-{[4-(2-fluorophenyl)phenyl]methyl}-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
N-[(4-methoxyphenyl)methyl]-3-(3-methyl-1H-pyrazol-1-yl)-N-{[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl}propanamide
3-benzoyl-1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
[2-(3-methoxyphenyl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]benzonitrile
(2S,4R)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-hydroxypropanamido)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
(4aR,8aR)-4-(2-propyl-1,3-thiazole-4-carbonyl)-octahydro-2H-1,4-benzoxazine
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-pyrrol-1-yl)pentan-1-one
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[(6-methylpyridin-2-yl)methyl]pyridin-2-amine
1-(cyclopropanesulfonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{2-[(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-(1-carbamoylcyclopentyl)-2-methyl-1,3-thiazole-4-carboxamide
5-tert-butyl-2-(1,3-thiazol-2-yl)-1H-1,3-benzodiazole
1-[(4-chlorophenyl)methyl]-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
4-[2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-fluoropyrimidin-4-yl]morpholine
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrimidine-5-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-{2-[(cyclopropylmethyl)sulfanyl]acetyl}pyrrolidine-3-carboxylic acid
methyl 2-(azepane-1-sulfonyl)-6-(cyclohex-3-ene-1-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-methyl-6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,3-benzothiazol-2-amine
2-amino-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
methyl 2-({1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)-1,3-oxazole-4-carboxylate
N-[(3S,4R)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-[3-(furan-2-yl)phenyl]-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
3-(furan-2-yl)-1-methyl-5-(2-phenoxyethyl)-1H-1,2,4-triazole
7-(pyridin-3-yl)-4-(1,3-thiazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-hydroxybenzamide
N-benzyl-N-methyl-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-methylacetamide
(3R,4S)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-3,4-dimethylpiperidin-4-ol
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine-2-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)acetamide
2-(4-methyl-6-{[2-(1,3-thiazol-4-yl)ethyl]amino}pyrimidin-2-yl)phenol
6-(morpholin-4-yl)-N4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidine-2,4-diamine
1-[(3aS,6aS)-5-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-octahydropyrrolo[3,4-b]pyrrol-1-yl]-2-methoxyethan-1-one
1-[4-(benzyloxy)piperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
3-{5-[(2-ethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-{[3-oxo-4-(2-phenylphenyl)piperazin-1-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(furan-2-yl)ethane-1,2-dione
4-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-2-amine
3,5-dimethoxy-N-({1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}methyl)benzamide
2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]-N,N-dimethylethane-1-sulfonamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-decahydro-2,7-naphthyridin-4a-ol
2-{3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}acetamide
3-{3-[5-(pyrrolidine-1-carbonyl)furan-2-yl]phenyl}-1H-pyrazole
3-methoxy-1-(5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperidine