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N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
1-methyl-3-(2-methylpropyl)-8-{[4-(2-methylpropyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]methanol
2-(2,4-dioxo-1,3-thiazolidin-3-yl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
(4aS,8aR)-1-(3-aminopropyl)-6-(quinolin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-fluoro-N-[4-(4-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
{4-[(1-cyclopentanecarbonylpyrrolidin-3-yl)methyl]phenyl}methanol
N-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}propanamide
4-({4-methyl-5-[1-(pyridine-2-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-[3-(1H-indol-2-yl)phenyl]-1-propanoylpyrrolidine-2-carboxamide
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}propan-1-one
(2E)-N-{[3-methyl-7-(2-oxo-2-phenylacetyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
6,7-dimethyl-4-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-2H-chromen-2-one
8-[2-(difluoromethoxy)benzoyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
3-(2-propyl-1H-imidazol-1-yl)quinoline
3-(morpholine-4-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[3-(2-chloro-6-methoxyphenyl)phenyl]methyl}cyclopropanamine
N-[(3-hydroxypyrrolidin-3-yl)methyl]-3-[4-(methylsulfamoyl)phenyl]propanamide
5-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
3-[5-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
1-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
3-methyl-8-[2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aS,8aR)-6-(4-cyclopentylpyrimidin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-phenyl-1-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]ethan-1-one
9-[(2R)-2-amino-2-phenylacetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-{2-[2-(trifluoromethyl)phenyl]ethyl}acetamide
7-{[(2-ethoxypropyl)(methyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-ethyl-8-(2-methylpropyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-{[(2E)-4-methylpent-2-en-1-yl]amino}-5-[(propan-2-yl)sulfamoyl]benzamide
4-(1-{furo[3,2-c]pyridin-4-yl}azetidin-3-yl)pyridine
(4aS,8aR)-6-[2-(propan-2-yl)pyrimidine-4-carbonyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(oxolane-2-carbonyl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
2-{4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1-methylpiperazin-2-yl}ethan-1-ol
2-[3-(methylsulfanyl)propanoyl]-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
2-(1-{[1-(6-methylquinoline-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
2-[2-(2-chlorophenoxymethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-(2-fluorophenyl)-4-{4-[(3-hydroxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}piperidin-4-ol
3-methyl-7-[2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(cyclopropylmethyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}-4-methoxypiperidine
6-butyl-2-(4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(1S,6R)-9-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
1-(1'-{6-[ethyl(methyl)amino]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)-2-methoxyethan-1-one
4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
N-[4-({[1-(ethoxymethyl)cyclobutyl]methyl}carbamoyl)phenyl]-2-methylfuran-3-carboxamide