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N-benzyl-2-chloro-4-acetamido-N-(3-hydroxy-2-methylpropyl)benzamide
3-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
2-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
(3-{3-[3-(2,5-dimethylpyrimidin-4-yl)phenyl]-1H-pyrazol-1-yl}propyl)dimethylamine
2-hydroxy-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
4-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyrimidin-2-amine
4-benzyl-3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)piperazin-2-one
3-(4-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
5-(1H-imidazol-1-yl)-2-(pyridin-3-yl)-1,3-benzoxazole
5-cyclopropyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,3,4-oxadiazol-2-amine
N-[1-(hydroxymethyl)cycloheptyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
6-ethyl-N-[3-(1H-indol-1-yl)propyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[4-(propan-2-yl)pyrimidin-2-yl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-3-(pyridin-3-yl)propanamide
N-[2-({1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidin-3-yl}formamido)ethyl]acetamide
(3aR,6aR)-2-(ethylcarbamoyl)-5-[(5-methylfuran-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-methyl-4-[3-(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyridine
4-{5-[1-(2-methylpropyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-[(1-phenylcyclopentyl)methyl]acetamide
4-{[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]sulfonyl}benzoic acid
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[2-(1H-pyrazol-1-yl)ethyl]amine
8-methoxy-2-methyl-5-[6-(propan-2-yl)pyrimidin-4-yl]quinoline
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxypyridine-3-carboxamide
4-{[4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinoline
3-{[1-benzyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
3-(3-methoxyphenyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
2-(1-benzyl-1H-pyrazol-4-yl)-N,N-dimethylquinoline-4-carboxamide
1-(2-methoxyacetyl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
(1R,3S)-7-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[1-(1H-imidazol-1-yl)propan-2-yl]amine
2-[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]-6-methylpyridine-3-carbonitrile
4-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
6-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}pyrimidin-4-amine
2-(1H-pyrazol-1-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}butanamide
2-{[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
N-(2-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-[(naphthalen-1-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
[(2,2-dimethyl-1-phenylcyclopropyl)methyl](methyl)(pyridin-4-ylmethyl)amine
4-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide
1-(2-benzylphenyl)-3-[2-(4-hydroxypiperidin-1-yl)ethyl]urea
7-cyclopentyl-2-(pyridin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
methyl 6-(2-{[2-(cyclohex-1-en-1-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
2-[1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-(4-methylpiperazin-1-yl)propan-1-one
4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-methyl-N-[2-(4-methylphenyl)propan-2-yl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide