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2-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
1-{2-[2-(3-methoxyphenyl)acetamido]ethyl}-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyrazolo[1,5-a]pyridine-2-carboxamide
8-(2,1,3-benzoxadiazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(2,2-diphenylethyl)-4-[2-(1H-pyrazol-4-yl)ethyl]morpholine
N-ethyl-3-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]sulfonyl}-N-(2-methylprop-2-en-1-yl)benzamide
1-cyclopentyl-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
(1S,5R)-6-benzyl-3-[3-(4-hydroxyphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1,2,3,4-tetrahydroisoquinoline
4-(5-methylfuran-2-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]benzamide
1-benzyl-N3-ethyl-4-oxo-N5-(2-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]pyridin-2-amine
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
(1R,2S)-N1-tert-butyl-N2-[3-(propan-2-yloxy)propyl]cyclohexane-1,2-dicarboxamide
{3-[(2-fluorophenyl)methyl]-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl}methanol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
4-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
(3S,4R)-3-ethyl-4-methyl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-4-ol
1-methyl-1-[1-(1,2-oxazol-3-yl)ethyl]-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
8-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-fluoro-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzene-1-sulfonamide
5-(5-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)-1H-1,3-benzodiazole
4-chloro-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-1H-pyrazole-3-carboxamide
(2S,4S)-4-(2-chlorobenzamido)-N-ethyl-1-[(3E)-pent-3-enoyl]pyrrolidine-2-carboxamide
2-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[(3-fluorophenyl)methyl]-N-[2-(4-methylphenyl)propan-2-yl]-6-oxopiperidine-3-carboxamide
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-acetamidopyrrolidine-1-carboxamide
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
(4aR,7aS)-1-(2-methoxyethyl)-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(2-hydroxyphenoxy)ethan-1-one
2-[2-(benzyloxy)phenyl]-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-(cyclohex-1-en-1-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-methyl-N-(naphthalen-1-ylmethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N,4-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1,3-thiazole-5-carboxamide
1'-(5-ethyl-2-methylpyrimidin-4-yl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[2-(benzyloxy)phenyl]pyrazine-2-carbonitrile
4-(1-ethyl-1H-pyrazole-4-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-(5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-(dicyclopropylmethyl)-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]propanamide
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypropan-1-one
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)[(2-methyl-1,3-oxazol-4-yl)methyl]amine
6-[3-(2-ethylphenoxy)azetidin-1-yl]pyrimidin-4-amine
5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
1-{4-[({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)methyl]thiophen-2-yl}ethan-1-one
3-ethyl-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-5-methyl-1,2-oxazole-4-carboxamide
4-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]piperazine-2-carboxylic acid