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2-{4-[2-chloro-5-(1H-pyrazol-1-yl)benzamido]-3,5-dimethyl-1H-pyrazol-1-yl}acetic acid
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(oxane-4-carbonyl)piperidine
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}thiolan-3-amine
N-{1-[1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
methyl 1-(2-methoxyethoxy)-2-oxo-8-[2-(3-phenylpiperidin-1-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-3-(4-methylbenzenesulfonyl)propan-1-one
1-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[(2-fluorophenyl)methyl]piperidine
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-4-methylbenzene-1-sulfonamide
3-[(4-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)methyl]pyridine
6-(2,5-dimethylfuran-3-yl)-N-(2-hydroxyethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1S,5R)-6-(1-benzoxepine-4-carbonyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-(3-phenylpropyl)-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylate
2-methyl-4-(2-methylphenyl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazine
2-ethyl-6-methyl-4-oxo-N-(pyridin-4-ylmethyl)-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-(2,3-dihydro-1H-isoindol-2-yl)-N-[2-(morpholin-4-yl)ethyl]pyridine-2-carboxamide
1-{1-[2-(methylamino)acetyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butanamide
3-(3-hydroxy-3-methylbutyl)-N-[(1-hydroxycyclohexyl)methyl]benzamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-3-azaspiro[5.5]undecan-9-amine
7-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
6-(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4,4,4-trifluoro-1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}butan-1-one
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[4-(4-methylpiperazine-1-carbonyl)morpholin-3-yl]acetamide
2-(2-methoxyethoxy)-1-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]ethan-1-one
4,6-dimethyl-3-[4-(quinazolin-4-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(2-ethoxyethyl)-N-methyl-2-oxo-N-(pyrazin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(butylsulfanyl)-N4-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidine-4,6-diamine
3-{3-[1-(2-hydroxyethyl)-4-phenyl-1H-imidazol-5-yl]-1H-indol-1-yl}propanamide
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(3,4-dimethylphenyl)methyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-3-(2-ethylphenoxy)azetidine
4-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1-methylpyrrolidin-2-one
3-[1-(4-hydroxybutan-2-yl)piperidin-4-yl]-N-phenylpropanamide
4-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
7-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidine
2-amino-5-methyl-4-(3-methyl-1H-indol-2-yl)-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]naphthalene-1-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-[3-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl}ethan-1-ol
(3aS,6aS)-2-(1H-indol-7-ylmethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4S)-4-amino-N-ethyl-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidine-2-carboxamide
N-[(4-fluorophenyl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
3-{1-[1-(cyclohexylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
N-({3-methyl-7-[2-(phenylsulfanyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-phenylmethanesulfonamide
4-benzyl-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-ol
2-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}benzonitrile
N,N,4-trimethyl-5-[4-(9H-purin-6-yl)piperazine-1-carbonyl]pyrimidin-2-amine
1-(1H-imidazol-2-ylmethyl)-2-[2-(thiophen-2-yl)ethyl]piperidine