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1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-[2-(morpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
1-methyl-N-[2-(5-methylfuran-2-yl)ethyl]azepane-2-carboxamide
N-cyclohexyl-2-(3-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
3-hydroxy-2-[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propanoic acid
1-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-4-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-(furan-2-ylmethyl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidine-1-carboxamide
8-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1-oxa-8-azaspiro[4.6]undecane
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-6-yl]oxy}acetamide
2-amino-N-[(1-benzylpiperidin-4-yl)methyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide
{[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}dimethylamine
N-cyclopropyl-4-{methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}pyridine-2-carboxamide
2-[(1R,3S,3aS,6aR)-1-(hydroxymethyl)-5-methyl-3-[3-(1H-pyrazol-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
3-{[2-(1-ethylpiperidin-4-yl)acetamido]methyl}-1,2,4-oxadiazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
4-{[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzonitrile
5-(4-methoxyphenyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}furan-2-carboxamide
N-butyl-3-ethynyl-N-(propan-2-yl)benzamide
N-[(3-chlorophenyl)methyl]-1-(cyclohexylmethyl)-6-oxopiperidine-3-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-6-methoxy-N-methyl-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[1-(2-phenylethyl)-4-(quinolin-4-ylmethyl)piperazin-2-yl]ethan-1-ol
2-[(4-chlorophenyl)methyl]-8-(2-methoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
2-[2-(1-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
{1-[1-(6-methoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
(isoquinolin-5-ylmethyl)({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-2-(1H-pyrazol-1-yl)acetamide
ethyl 4-{[(1R,2S)-2-[3-(1H-1,2,4-triazol-1-yl)propanamido]cyclobutyl]amino}piperidine-1-carboxylate
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(1S,5R)-6-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
3-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
3-[(3R,4S)-1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-(4-ethylpiperazin-1-yl)-3-[3-({[3-(pyridin-3-yl)propyl]amino}methyl)phenoxy]propan-2-ol
1-[7-acetyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
4-{[(4-methylphenyl)methyl]amino}-N-[1-(pyridin-4-yl)propan-2-yl]benzamide
4-({7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}methyl)benzene-1-sulfonamide
2-{[(1-ethyl-1H-imidazol-5-yl)methyl]amino}-N-[1-(4-methylphenyl)ethyl]acetamide
5-{[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl}-N-methylfuran-2-carboxamide
[4-(2-phenylethyl)-1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl]methanol
2-(3-fluorophenyl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
methyl 2-[4-(4-methylphenyl)-3-oxopiperazine-1-carbonyl]piperidine-1-carboxylate
1-methyl-4-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperazin-2-one
(3R,9aR)-3-(hydroxymethyl)-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[2-cyclopropyl-7-(5-fluoropyrimidin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}acetamide
1-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-3-(1H-indazol-4-yl)urea
1-phenyl-5-({4-propyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1H-pyrazole
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-chlorobenzamide
(1R,3S)-3-(2-aminoethoxy)-7-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-7-azaspiro[3.5]nonan-1-ol
6-cyclopropyl-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]pyrimidin-4-amine
2-(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethan-1-ol