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1,6-dimethyl-N-(1,3,4-thiadiazol-2-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carboxamide
4-(benzylsulfamoyl)-N-[(3R)-pyrrolidin-3-yl]benzamide
(3S,4R)-1-(1,1-dioxo-1λ6-thiane-4-carbonyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
7-fluoro-N-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-N-propylquinoline-4-carboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-3-carboxylate
N-(3,5-dimethylphenyl)-N'-(furan-2-ylmethyl)-N'-(pyridin-4-ylmethyl)propanediamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-ethyl-3-methyl-1H-pyrazole-4-sulfonamide
1-(4-methylphenyl)-4-[2-(oxan-2-ylmethoxy)acetyl]piperazin-2-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(furan-3-ylmethyl)acetamide
5-chloro-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-carboxamide
4,6-dimethyl-N-[2-(5-methylthiophen-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
6-(morpholin-4-yl)-N-[1-(thiophen-2-yl)propan-2-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(2S,4R)-4-amino-N,N-diethyl-1-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidine-2-carboxamide
N-cyclobutyl-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-2-carboxamide
(3S,5S)-5-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-1-methylpyrrolidin-3-amine
2-amino-4-(3,4-dihydroxyphenyl)-6-(1,2-dimethyl-1H-indol-3-yl)pyridine-3-carbonitrile
2-fluoro-6-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]benzamide
N-[2-methoxy-5-({[2-(pyridin-3-yloxy)propyl]carbamoyl}amino)phenyl]propanamide
propyl 4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-[(3,5-difluorophenyl)methyl]-8-(2-ethoxyethyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
3-(3-hydroxyquinoxalin-2-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
4-amino-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)pyridine-2-carboxamide
(1S,6R)-3-methyl-9-({2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
8-[(3-phenylphenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
2-amino-4-[2-(furan-2-yl)pyrimidin-5-yl]-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
(4aS,7aR)-1-(3-chloro-1H-indole-2-carbonyl)-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 5-[2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-(ethylsulfanyl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-(4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperazin-1-yl)acetamide
1,3,5-trimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1H-pyrazole-4-sulfonamide
4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}benzonitrile
N-(furan-3-ylmethyl)-5-{1-[(2-hydroxypyridin-4-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-(1H-imidazol-1-ylmethyl)-N-[2-(morpholin-4-ylmethyl)phenyl]piperidine-1-carboxamide
1-cyclohexyl-N3-cyclopropyl-4-oxo-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
3-(N-benzyl-1-2,3-dihydro-1H-inden-1-ylformamido)propanamide
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
(1S,5R)-3-(4-propylbenzoyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-4-amino-N-methyl-1-[(3E)-4-phenylbut-3-enoyl]pyrrolidine-2-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
(3S,4R)-1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-(hydroxymethyl)piperidin-3-ol
N-[2-(2-methoxyphenyl)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(2,6-difluorophenyl)methyl]-4-(2-phenylpropyl)-1H-1,2,3-triazole
8-fluoro-2-{[(oxolan-3-ylmethyl)amino]methyl}quinolin-4-ol
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
({4-ethyl-5-[1-(pyridazine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
6-oxo-N-[(3-phenylphenyl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-(1H-1,2,4-triazol-3-yl)benzamide