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3-(3-hydroxy-1,2-oxazol-5-yl)-1-(6-hydroxy-1,4-diazepan-1-yl)propan-1-one
3-(5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
(1S,5R)-6-(cyclobutylmethyl)-3-(2-methyl-6-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-6-(1,2-oxazole-3-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N'1-[(2-benzyl-1,3-thiazol-4-yl)methyl]cyclopropane-1,1-dicarboxamide
N-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-2-(2-fluorophenyl)ethyl}-N-methyl-3-(methylsulfanyl)propanamide
1-(cyclohexylmethyl)-N3-cyclopropyl-4-oxo-N5-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
benzyl 4-[2-(2,6-dioxo-1,3-diazinan-1-yl)acetyl]-1,4-diazepane-1-carboxylate
1-benzyl-5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
(4aS,8aR)-6-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
(2S,4R)-4-amino-1-(2,2-diphenylacetyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(1-methylpiperidin-2-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)acetamide
4-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-propyl-1,3-thiazole
6-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-N-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(4-{3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]pyridin-2-yl}phenyl)methanol
7-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenol
2-[(naphthalen-1-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
7-[(3-methylphenyl)methyl]-2-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decane
2-{4-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
(5-{1-[2-(2-chlorophenoxy)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
7-cyclopropanecarbonyl-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-ethyl-7-(2-methoxybenzamido)-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
2-({4-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]pyrimidin-2-yl}(methyl)amino)-N-methylacetamide
5-[(4-chloro-3-methyl-1H-pyrazol-1-yl)methyl]-3-cyclopropyl-1H-1,2,4-triazole
1-ethyl-3-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]piperidine
ethyl 4-({[1-(7-chloroquinolin-4-yl)-4-(ethoxycarbonyl)-1H-pyrazol-5-yl]methyl}amino)piperidine-1-carboxylate
ethyl 1-(cyclopropylmethyl)-5-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2-{1-[(4-methylphenyl)methanesulfonyl]piperidin-2-yl}ethyl)acetamide
N-{3-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propanamido]phenyl}-2-methoxybenzamide
N-(pyridin-3-ylmethyl)-3-[1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]propanamide
5-methyl-1-{2-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-6-(cyclopropylmethyl)-3-(quinoline-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)acetyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4S)-1-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-{3-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}methanesulfonamide
[(4aS,8aR)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridin-4a-yl]methanol
4-(2-{1-[(3-chloro-2-fluorophenyl)methyl]piperidin-2-yl}ethyl)morpholine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]pyridine-2-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(6-cyclopropylpyrimidin-4-yl)-6-methylquinoline
4-(azepan-1-yl)-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
[(2S,6S)-4-(pyridin-4-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(3aS,6aS)-5-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-methyl-octahydropyrrolo[2,3-c]pyrrole
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)(pyridin-2-ylmethyl)amine
4-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
6-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2,4-dimethylpyridine-3-carbonitrile
3-[2-(4-methylpentyl)morpholine-4-carbonyl]-1,2-dihydroquinolin-2-one
1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-3,4,4-trimethylpyrrolidin-3-ol
2-(2-aminoethyl)-N,5,6-trimethyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine