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N-(2-methoxyethyl)-3-({1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
N-methyl-2-oxo-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
6-{[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-amino-4-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-5-methyl-6-(pyridin-2-yl)pyridine-3-carbonitrile
ethyl 4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
4-benzyl-1-[2-(4-fluorophenoxy)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[2-(azepan-1-yl)ethyl](methyl)amino}-N-cyclopentylpropanamide
4-(1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-5-methylpyrimidine
N-(furan-2-ylmethyl)-7-[(3-methoxyphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
(3S,4R)-1-(1-ethylpiperidin-4-yl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-methoxy-4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
[(2S,6S)-4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
1-methyl-4-[3-(1H-pyrazol-4-yl)benzoyl]-1,4-diazepan-6-ol
2-cyclopentyl-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
1-cyclopentyl-5-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
methyl 3-[4-({1-ethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)-1H-pyrazol-1-yl]propanoate
4-({[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
(2S,4S)-4-amino-N,N-diethyl-1-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]pyrrolidine-2-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-2-(1,3-thiazol-4-yl)acetamide
N,N-dimethyl-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)benzamide
2-benzyl-8-{2-[methyl(phenyl)amino]acetyl}-2,8-diazaspiro[4.5]decan-3-one
2-(4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenyl)pyridine
5-(4-{[2,5-dimethyl-1-(pyridin-3-yl)-1H-pyrrol-3-yl]methyl}piperazin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl][(2E)-3-(furan-2-yl)prop-2-en-1-yl]methylamine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[(3,5-dimethoxyphenyl)methyl]piperidine
(2E)-1-[(4aR,8aS)-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-3-(2,4-difluorophenyl)prop-2-en-1-one
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-2-(ethylamino)pyrimidine-5-carboxamide
1-ethyl-5-(4-methanesulfonyl-1,4-diazepan-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-methylpropyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-(3-phenoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
3-cyclopropyl-6-(2,3-dihydro-1H-inden-1-ylmethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N,N-dimethyl-5-[(5-methylfuran-2-yl)methyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[1-cyclohexyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
1-[(1-{6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
(2S,4S)-N-ethyl-1-(3-methylbut-2-en-1-yl)-4-[4-(methylsulfanyl)benzamido]pyrrolidine-2-carboxamide
4-phenyl-N-(2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1H-imidazole-5-carboxamide
1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-methyl-1-{1-[6-(thiomorpholin-4-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
6-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}({[2-(prop-2-en-1-yloxy)phenyl]methyl})(pyridin-4-ylmethyl)amine
3-cyclohexyl-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-(5-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
[(1-ethyl-1H-pyrazol-4-yl)methyl][(2-methyl-1H-imidazol-4-yl)methyl](2-methylpropyl)amine