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1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
3-(2,5-dimethoxyphenyl)-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine
(4aR,7aS)-1-acetyl-4-[(4-chlorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4R)-4-(hydroxymethyl)-1-[5-(propan-2-yl)thiophene-3-carbonyl]piperidin-3-ol
1-{1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}-4-phenylpiperazine
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
(2S)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}butanamide
1-{1H-pyrrolo[2,3-b]pyridin-6-yl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(dimethylamino)-N-ethyl-2-(2-methylphenyl)-N-(oxan-4-ylmethyl)acetamide
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(3-fluorophenyl)methyl]pyrrolidine-2-carboxylate
1-{5-cyclopropyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
ethyl 3-[(3-chlorophenyl)methyl]-1-(prop-2-ene-1-sulfonyl)piperidine-3-carboxylate
[(3R,4R)-1-(3,4-difluorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(3S,4R)-1-(cyclopentylcarbamoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
3-{imidazo[1,2-a]pyridin-2-yl}-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}propan-1-one
1-{4-[1-(2-fluorophenyl)cyclopropanecarbonyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
4-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1,2-dihydroquinazolin-2-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]acetamide
N-methyl-3-[methyl({[2-(5-methylfuran-2-yl)phenyl]methyl})amino]butanamide
2-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[4-(4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}piperidin-1-yl)phenyl]-5-phenylpentanamide
1-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-propylurea
methyl 3-[3-(2-{methyl[2-(pyridin-2-yl)ethyl]carbamoyl}ethyl)piperidine-1-carbonyl]benzoate
(2S)-2-[3-(cycloheptylcarbamoyl)propanamido]-3-(4-hydroxyphenyl)propanoic acid
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-4-methylpyrimidin-2-amine
6-fluoro-3-(oxan-2-ylmethyl)-3,4-dihydroquinazolin-4-one
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
2-(dimethylamino)-7-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(1-methyl-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
(3S,4R)-1-[3-(difluoromethoxy)benzoyl]-4-methylpiperidine-3,4-diol
N-[1-(ethylsulfanyl)propan-2-yl]-1-(3-methylphenyl)piperidin-4-amine
6-ethyl-3-[1-(2-hydroxyethyl)-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]-1,5-dimethyl-1,2-dihydropyridin-2-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
2-hydroxy-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)pyridine-3-carboxamide
5-(3-methoxypyridin-2-yl)-1,2,3,4-tetrahydroisoquinoline
(1R,3S)-3-methoxy-7-[5-(methoxymethyl)thiophene-2-carbonyl]-3-methyl-7-azaspiro[3.5]nonan-1-ol
4-(1-ethyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5,6-dimethyl-3-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
1-cyclopentyl-N5-[3-(dimethylamino)-2,2-dimethylpropyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3,4,4-trimethyl-1-[2-(morpholin-4-yl)benzoyl]pyrrolidin-3-ol
7-(cyclopropylmethyl)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-(1-benzofuran-2-yl)-3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-1,2,4-triazine
2-hydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}benzamide
(3S,4R)-1-[2-methyl-2-(piperidin-1-yl)propyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-ethyl-2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide