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2,2,2-trifluoro-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}ethane-1-sulfonamide
N-[(4-hydroxyazepan-4-yl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}-7-methyl-3,4-dihydroquinazolin-4-one
2-(dimethylamino)-2-(4-methylphenyl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
N-phenyl-3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
N-[2-hydroxy-2-(3-phenoxyphenyl)ethyl]-4-methylpiperidine-4-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one
(2R,6S)-4-[1-(5-chloro-3-fluoropyridin-2-yl)piperidin-4-yl]-2,6-dimethylmorpholine
7-[(2,3-difluorophenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-methoxy-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
4-(5-acetylthiophene-3-carbonyl)-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
5-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole
2-{2-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-oxoethoxy}acetamide
N-(2-methoxyethyl)-1-{1-[2-(pyridin-2-yl)ethyl]piperidin-4-yl}piperidine-3-carboxamide
7-cyclobutanecarbonyl-2-methyl-N-(thiolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(pyridin-3-ylmethyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[(2,5-dimethylphenyl)methyl]-1,4-diazepan-5-one
N-[2-(methylamino)ethyl]-3-[(1-phenylcyclopropyl)sulfamoyl]benzamide
N-ethyl-3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclohexanecarboxamide
N,3-dimethyl-1-propyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
4-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-methoxy-4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-(furan-3-yl)-4-phenyl-1H-imidazole
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-[(2,3-dichloro-6-fluorophenyl)methyl]-4,4-dimethylpyrrolidin-2-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-(2-methylpropyl)-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide
(3R,4S)-4-cyclopropyl-1-(5-ethyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-amine
N-({5-[3-(methylsulfanyl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-(pyridin-2-yl)-N-(trimethyl-1H-pyrazol-4-yl)piperazine-1-carboxamide
2-(2-{[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}ethyl)-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-[3-(piperidine-1-carbonyl)phenyl]-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
5-ethyl-4-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}pyrimidin-2-amine
2,3-dimethyl-7-{2-[(propan-2-yl)amino]benzoyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
[(3-chloro-5-fluorophenyl)methyl](methyl)[1-(pyridin-4-yl)ethyl]amine
ethyl 1-[(6-chloroquinolin-2-yl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
methyl 4-{4-[5-(2-methylbenzamido)-1H-pyrazol-1-yl]piperidin-1-yl}-4-oxobutanoate
3-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)benzamide
3-{1-[(3-cyanophenyl)methyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
4-methyl-3-({2-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-4H-1,2,4-triazole
2-(2,4-dimethoxyphenyl)-1H-1,3-benzodiazole-5-carbonitrile
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[4-(furan-2-yl)phenyl]-1-(3-phenoxypropanoyl)piperidine-3-carboxamide
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyrazin-2-yl)propan-2-yl]pyridin-2-amine
5-(azepane-1-carbonyl)-N-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-(2,3-difluorophenoxymethyl)-N-ethyl-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one