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N-(2-methyl-1-{3-methyl-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}propyl)acetamide
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)(quinoxalin-2-ylmethyl)amine
1-{3-[3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
2-{1-[(5-propylfuran-2-yl)methyl]azetidin-3-yl}pyridine
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-5-one
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2-(thiophen-3-yl)acetamide
2-{[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-1-(4-hydroxyphenyl)ethan-1-one
1-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-4-phenylpiperidin-4-yl]ethan-1-one
1-(1-methylpiperidin-4-yl)-4-[3-(trifluoromethyl)benzoyl]piperazine
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(1,2-oxazol-3-ylmethyl)pyrimidine-5-carboxamide
2-methoxy-N-{[1-(pent-2-yn-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}acetamide
1-(cyclohexylmethyl)-4-oxo-5-[4-(piperidin-1-yl)piperidine-1-carbonyl]-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-benzyl-3-ethyl-1-(1,8-naphthyridine-2-carbonyl)-1,4-diazepan-5-one
2-{5-[2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-N-(propan-2-yl)acetamide
2-(1H-1,3-benzodiazol-1-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(3-methoxyphenyl)piperazine
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-(pyrimidin-4-ylmethyl)benzamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-methoxyphenyl)methyl]-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
1-(2,2-dimethylpropyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}acetamide
2-(2-{1-[2-(5-acetylthiophen-3-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(4-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}piperidin-1-yl)butan-1-one
5-tert-butyl-4-{[2-(trifluoromethyl)morpholin-4-yl]methyl}furan-2-carboxamide
(5S,9aS,9bS)-5-(2,1,3-benzoxadiazol-4-yl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-(morpholin-4-ylmethyl)-1,4-oxazepane
5-[1-(2,2-dimethyloxane-4-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N,N-dimethylpyridine-3-carboxamide
1-(4-{4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}piperidin-1-yl)ethan-1-one
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)propanamide
1-(3-methylphenyl)-4-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]pyrrolidin-2-one
5-{2-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}-2-methoxy-6-(prop-2-en-1-yl)phenol
2-(2-hydroxyethyl)-9-[(2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]pyrimidin-4-yl}piperidin-4-ol
3-methyl-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pentanamide
8-(1-benzofuran-2-ylmethyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{[5-(7-hydroxy-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)furan-2-yl]methyl}-N-methylmethanesulfonamide
N-cyclopropyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]-1,3-thiazole-5-carboxamide
methyl 2-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}benzoate
1-(2-benzylphenyl)-3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]urea
8-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[benzyl(methyl)amino]-3-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide
3-{[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
(3S,9aR)-8-[(3,4-difluorophenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-7,8-dimethyl-2-(2-methylpyrimidin-5-yl)-N-(propan-2-yl)quinoline-4-carboxamide