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5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(3-methoxypropyl)-1H-pyrazole-4-carboxamide
2-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-[N-cycloheptyl-1-(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]acetic acid
(4aS,8aR)-6-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}pyridin-2-amine
7-(3-chlorothiophene-2-carbonyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-(methoxymethyl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyrimidin-4-amine
3-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-pentylpiperidine-1-carboxamide
(3S,4R)-3-[(dimethylsulfamoyl)amino]-N-(2-phenylethyl)-4-(propan-2-yl)pyrrolidine-1-carboxamide
3-[4-(4-methoxyphenoxy)piperidin-1-yl]-6-methylpyridazine
N-ethyl-15-methyl-13-oxo-N-(pyridin-4-ylmethyl)-9-(thiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
1-[(3aS,6aS)-5-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)-octahydropyrrolo[3,4-b]pyrrol-1-yl]-2-methoxyethan-1-one
4-{[5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-amine
2-methoxyethyl 4-[(3-fluorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
3-methyl-N-({1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidin-3-yl}methyl)but-2-enamide
3-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
2,2-dimethyl-6-[3-(phenylamino)piperidine-1-carbonyl]-3,4-dihydro-2H-pyran-4-one
(1R,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
{1-[3-(azocane-1-sulfonyl)benzoyl]pyrrolidin-3-yl}methanamine
2-{[5-(2-amino-6-tert-butyl-3-cyano-5,6,7,8-tetrahydroquinolin-4-yl)pyrimidin-2-yl]amino}acetic acid
1-{5-[(cycloheptylamino)methyl]-2-methoxyphenoxy}-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
N-cyclopropyl-6-(dimethylamino)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide
3-(3-methoxyphenyl)-5-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-{2-[4-(pyridin-4-yl)piperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-(3-methylpiperidin-1-yl)-3-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}propan-1-one
5-methyl-N-(3-methylbutyl)-4-(piperidin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-{4-[(3S,4S)-4-hydroxy-1-(4-methoxybenzoyl)pyrrolidin-3-yl]-1,4-diazepan-1-yl}ethan-1-one
4-{1-butyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
3-methyl-4-[3-(propan-2-yl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]pyridine
N-methyl-N-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}oxolan-3-amine
1-(3-methoxypropyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3S,9aR)-3-(cyclohexylmethyl)-8-(2,4,5-trifluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
4-(2-oxo-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)piperazin-2-one
7-(cyclopropylmethyl)-2-[(3-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-(1H-pyrazol-3-yl)benzamide
2,5-dimethyl-N-[2-(pyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-ethyl-4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methyl-1,2-oxazole
1-(2-methyl-1-benzofuran-5-carbonyl)-4-[(methylsulfanyl)methyl]piperidine
N-(3-chloro-4-methoxyphenyl)-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}propanamide
2-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
3,7-dimethyl-8-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}-2,3,6,7-tetrahydro-1H-purine-2,6-dione
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(2-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
(3S,4R)-3-ethyl-4-methyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-ol
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-{[(3R)-pyrrolidin-3-yl]sulfamoyl}benzamide
3-{1-[(3-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-1-[(1S,2S)-2-hydroxycyclohexyl]urea
5-(3-{[(1,3-benzoxazol-2-yl)amino]methyl}pyrrolidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one