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1-ethyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
5-{[2-(3-phenylpiperidin-1-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
6-methyl-2-[(4-methyl-1H-imidazol-5-yl)methyl]-5-[5-(pyridin-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-4-ethyl-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-[8-(trifluoromethyl)quinolin-4-yl]piperidin-3-ol
N,N-dimethyl-4-(1-{[(2-methyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-indazol-5-yl)benzamide
4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(4aR,8aR)-7-{[3-(furan-2-yl)phenyl]methyl}-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
[(2S,4R)-1-(1-benzofuran-2-ylmethyl)-4-(dimethylamino)pyrrolidin-2-yl]methanol
1-(cyclopropylmethyl)-5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-fluoro-2-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,4-dihydroquinolin-4-one
1-cyclopropyl-4-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}pyrrolidin-2-one
2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carbonitrile
1-benzyl-N,N-dimethyl-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4-(4-methoxybenzoyl)piperazine
3,4,7-trimethyl-2-(3-phenylpiperazine-1-carbonyl)-1H-indole
3-[5-(ethanesulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-2-methyl-6-(trifluoromethyl)pyridine
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-(2-methoxyphenoxy)azetidine
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
8-{1-[3-(morpholin-4-yl)propyl]-1H-imidazol-2-yl}quinoline
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-[(2S)-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carbonyl]piperidine
1-[(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
7-methyl-4-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
(1R,7S)-3-(2-ethoxyethyl)-6-(4-ethylpiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[2-methyl-4-({2-[(pyridin-3-yl)amino]ethyl}amino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
4-methyl-N-{4-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl]phenyl}-3-oxopiperazine-1-carboxamide
1-(4-fluorophenyl)-3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
methyl 3-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
4-[(2-{4-oxo-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-2-yl}phenyl)methyl]-3-(propan-2-yl)piperazin-2-one
2-(adamantan-1-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-{3-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]propyl}-3,4-dihydroquinazolin-4-one
N-methyl-2-(pyridin-2-yl)-N-(1,3-thiazol-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
(2S,4R)-4-amino-N-[2-(4-methoxybenzenesulfonamido)ethyl]pyrrolidine-2-carboxamide
N-[3-(4-{[2-(morpholin-4-yl)ethyl]amino}piperidin-1-yl)phenyl]-4-phenylbutanamide
N-{2-[5-(3-fluoro-2-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}propane-1-sulfonamide
(2R)-2-cyclohexyl-2-hydroxy-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]acetamide
N-(2-hydroxyethyl)-1-(4-methoxyphenyl)-2,2-dimethyl-N-(1,3-thiazol-2-ylmethyl)cyclopropane-1-carboxamide
4-ethyl-1-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-diazepan-5-one
1-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}pyrrolidin-2-one
1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-[methyl(propan-2-yl)amino]ethan-1-one
ethyl 4-{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}piperazine-1-carboxylate
N-[2-(ethanesulfonyl)ethyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
5-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
2-{[2-(2-methylphenyl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
1-(2,3,5,6-tetramethylbenzoyl)-2,5-dihydro-1H-pyrrole