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3-(4-chlorobenzoyl)-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine
4-[({thieno[2,3-d]pyrimidin-4-yl}amino)methyl]-1,3-thiazol-2-amine
6-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
4-(2-methoxyphenoxy)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
4-(1,3-benzothiazol-2-yl)-1-(pyridin-2-ylmethyl)piperazine-2-carboxylic acid
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
2-(dimethylamino)-2-(3-fluorophenyl)-N-(3-hydroxypropyl)acetamide
3-{1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
dimethyl({3-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}methyl)amine
N-[3-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)carbamoyl}amino)phenyl]-2-methoxyacetamide
3-(3-chlorophenyl)-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3-phenylpropanamide
N-ethyl-N-methyl-2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
1-[2-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
(4aS,7aR)-1-[(3-methoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-{1-[(2-fluorophenyl)methyl]-4-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-(3-fluorophenyl)-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(trimethyl-1H-pyrazol-1-yl)acetamide
1-{2-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
1-[7-(cyclobutylsulfamoyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]cyclopropane-1-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[2-(dimethylamino)ethyl]-8-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,9R)-6-oxo-N-[3-(1H-1,2,4-triazol-1-yl)phenyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carboxamide
2-methyl-3-[4-(pyrrolidine-1-sulfonyl)phenyl]-6-(4H-1,2,4-triazol-4-yl)pyridine
5-methyl-1-propyl-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
2-[(3-methoxyphenyl)methyl]-8-(pyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,6-dimethyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-{3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]phenyl}pyrrolidin-2-one
N-(4-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}phenyl)acetamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-2-(1H-imidazol-1-yl)acetamide
2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-N-methylbutanamide
N-[(5-methylpyrazin-2-yl)methyl]-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
methyl 9-(cyclopentyloxy)-3-(3-fluoro-4-methoxybenzoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(4-methylpiperidine-1-carbonyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine
4-(4-chlorophenyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]butanamide
N,4-dimethyl-4-[(2,3,6-trimethylquinolin-4-yl)formamido]pentanamide
2-(1-ethylpiperidin-4-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]acetamide
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbenzamide
4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
N-methyl-2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-[1-(pyridin-2-yl)ethyl]acetamide
6-[1-(1H-1,3-benzodiazol-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-methyl-5-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(4aR,7aS)-1-(cyclopropylmethyl)-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 2-{N-methyl-2-[N-(3-methylphenyl)methanesulfonamido]acetamido}acetate
4-{1-[1-methyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]cyclohexyl}morpholine
4-methoxy-6-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]pyrimidine
4-[3-(2-methoxyethyl)-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
[4-(2,3-dihydro-1H-isoindol-2-yl)quinazolin-2-yl]methanol
2-(4-amino-3-fluorophenyl)-2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)acetic acid