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(2S,4S)-4-[(1-benzylpiperidin-4-yl)amino]-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-methyl-2-[methyl(piperidin-4-yl)amino]-N-[2-(pyridin-2-yl)ethyl]acetamide
7-fluoro-3-[(2-{2-[(propan-2-yl)amino]pyrimidin-5-yl}-1H-imidazol-1-yl)methyl]-1,2-dihydroquinolin-2-one
1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
4-[(1-methoxypropan-2-yl)amino]-5-methyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[3-(4-fluorophenoxy)piperidin-1-yl]acetamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-methylphenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-methyl-4-({4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazin-1-yl}methyl)phenol
N-(2-methylpropyl)-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
2-{1-[2-(1H-imidazol-2-yl)phenyl]-N-methylformamido}-N-methylpropanamide
2-methyl-N-[(3S)-2-oxoazepan-3-yl]-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-1,3-thiazole-4-carboxamide
(2R,3R)-3-amino-1'-(quinoline-8-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
{3-[(4-fluorophenyl)methyl]-1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-yl}methanol
(2R,3S,6R)-5-(1H-indole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]azocane
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,2,3-triazole
3-(4-chlorophenyl)-5-(3-fluoro-4-methoxybenzoyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N,N-dimethylacetamide
(1S,6R)-9-[2-(propan-2-yl)pyrimidine-4-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
(5-{[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
2-{4-[(5-methylfuran-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
ethyl 4-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetyl}piperazine-1-carboxylate
1-[(4-methoxypiperidin-1-yl)sulfonyl]-2-(2-phenylethyl)piperidine
N-(2-methoxyethyl)-3-(2-methyl-1H-indol-1-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
3-[4-(4-hydroxypiperidin-1-yl)piperidine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
6-tert-butyl-N,1-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[4-(1-acetylpiperidine-4-carbonyl)piperazin-1-yl]-2-(naphthalen-1-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
methyl 2-{[3-(benzylamino)-5-(phenylsulfamoyl)phenyl]formamido}acetate
2-(1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl)acetic acid
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(naphthalen-1-yl)ethan-1-one
3-(furan-2-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-7-chloro-4-hydroxy-N-methylquinoline-3-carboxamide
1-{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}imidazolidine-2,4-dione
5-{2-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,4R)-3-cyclopropyl-1-(3-methoxypyrazin-2-yl)-4-methylpyrrolidin-3-ol
4-[2-(2,3-dihydro-1H-inden-1-yl)acetamido]oxane-4-carboxylic acid
(1R,7S)-6-(4-ethylpiperazine-1-carbonyl)-3-[(3-methoxyphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(1S,5R)-3-[3-(1H-indol-3-yl)propanoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{4-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]piperazin-1-yl}-N-tert-butylacetamide
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-phenylbutane-1,4-dione
4-(4-fluorophenyl)-1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperidin-4-ol
3-(1-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazol-4-yl)benzonitrile
3-[4-(1-benzylpiperidin-4-yl)piperazin-1-yl]-6-chloropyridazine
1,3-dimethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3S,4R)-3-methoxy-1-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carbonyl]piperidin-4-amine
[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)(thiophen-2-ylmethyl)amine
(2S,4S)-4-benzamido-N-ethyl-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
(3R)-1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
2-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol