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N-[(2-chloro-6-fluorophenyl)methyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
(1S,4S)-2-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)-2-azabicyclo[2.2.1]heptane
2-[1-methyl-4-(1-methyl-1H-pyrrole-2-carbonyl)-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
1-{4-[(2-chloro-6-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(morpholin-3-yl)ethan-1-one
2-amino-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-6-(2-methylpropyl)pyrimidine-4-carboxamide
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
3-methyl-1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3-phenylpiperidine
5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-1-phenyl-1H-pyrazole
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxylate
4-hydroxy-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-[(1S,2S)-2-hydroxycyclohexyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-chloro-4-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenol
3-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}pyrazine-2-carbonitrile
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N4-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-methoxy-4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]pyridine
(3S,4R)-1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-ethyl-1-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]pyrrolidine-3-carboxamide
7-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(1H-imidazol-2-yl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidine
4-(5,6-dimethylpyrimidin-4-yl)-2-(6-methoxynaphthalen-2-yl)morpholine
5-acetyl-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-1-{[3-(difluoromethoxy)phenyl]methyl}urea
4-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidine-1-sulfonamide
N-[2-(3,5-dimethoxyphenyl)-2-hydroxyethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
6-(2-fluoro-4-methoxyphenyl)-7-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[4-(benzyloxy)butyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(1R,5R)-6-(pyridin-2-ylmethyl)-3-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(2-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]-1H-pyrazole
4-[2-(4-phenyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-[4-(3-fluorophenyl)phenyl]-1-[2-(pyridin-2-yl)acetyl]piperidine-3-carboxamide
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N,5-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]thieno[2,3-d]pyrimidine-6-carboxamide
(3S,5R)-1-[(4-ethylphenyl)methyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-(1,4-oxazepane-4-carbonyl)-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
3-cyano-5-fluoro-N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)benzamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[(2-methoxyphenyl)methyl]piperidine
N-(1H-indol-2-ylmethyl)-4-pentanamidobenzamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-4-oxo-4H-chromene-2-carboxamide
3-(cyclopropylsulfamoyl)-5-(1H-pyrazol-4-yl)benzoic acid
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
2-(4-chlorophenoxy)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-cyclohexyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(cyclopropylmethyl)-4-(1,2-oxazole-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-[1-(morpholin-4-ylmethyl)cyclopentyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
[(2,2-dimethyloxan-4-yl)methyl](methyl)(quinolin-8-ylmethyl)amine
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(2,4-dimethoxyphenyl)methyl]piperazin-2-one