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3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}urea
3-(azetidine-1-carbonyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]benzene-1-sulfonamide
3-({4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]piperidin-1-yl}methyl)phenol
5-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-1,2,4-triazole
(4aR,7aS)-1-acetyl-4-[1-(4-methylphenyl)cyclopropanecarbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S)-1-{[5-(5-chlorothiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3-fluoropyrrolidine
6-fluoro-2-({[3-(methylsulfanyl)propyl]amino}methyl)quinolin-4-ol
1-(furan-2-ylmethyl)-3-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}urea
1-ethyl-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}benzamide
1-(2-{1-[3-(3,5-dimethylphenyl)propanoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
4-[(4-methyl-5-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
(1S,6R)-3-(piperidine-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
5-methyl-N-({3-methyl-7-[(2E)-3-phenylprop-2-en-1-yl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)pyrazine-2-carboxamide
N-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-2-methylpropanamide
1-[(4-phenylphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
ethyl 3-(2-methoxyethyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
4-(4-chlorophenoxy)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-ethyl-N-methyl-N-(1-methylpiperidin-4-yl)piperidin-3-amine
3-(2-chloro-6-methoxyphenyl)-5-methylpyridin-2-amine
5-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-4-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(3S,5R)-1-benzoyl-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
4-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N,N-dimethyl-4-oxobutanamide
4-[4-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
2-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-6,7-dimethyl-1H-1,3-benzodiazole
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)pent-4-enamide
2-(2-chlorophenyl)-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-hydroxyethan-1-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-[3-(dimethylamino)propyl]-5-(furan-2-yl)-N-methyl-1H-pyrazole-4-carboxamide
N-(3-hydroxypropyl)-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
2-(hydroxymethyl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
(2S,4S)-N-ethyl-4-[3-(4-methyl-1H-pyrazol-1-yl)propanamido]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
6-(2-chlorophenyl)-N-ethyl-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[(4-fluorophenyl)methyl]-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[4-(2-fluorophenoxy)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
4-(8-methoxy-2H-chromen-3-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
5-acetyl-N-cyclopropyl-N-(1H-indol-5-ylmethyl)thiophene-3-carboxamide
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-(3-methoxypropyl)piperidine-3-carboxamide
2-amino-6-cyclopropyl-4-(3,4-dimethoxyphenyl)pyridine-3-carbonitrile
8-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
N-benzyl-6-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
6-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}quinoxaline
2-amino-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-4-carboxamide
5-(1H-indol-1-ylmethyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]furan-2-carboxamide
3-[1-benzyl-2,4-dioxo-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]propanamide
1-{2-methoxy-5-[(4-methylpiperazin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
N-(1-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
(2S)-2-amino-2-cyclohexyl-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one