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N-[(3R,4R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
(3S,4S)-1-(6-chloro-1,3-benzothiazol-2-yl)piperidine-3,4-diol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-2-hydroxy-N-(2-methoxyethyl)-6-methylpyridine-3-carboxamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidine
9-methoxy-7-(2-methylphenyl)-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-[4-(5-methyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]-9H-purine
2-(ethylamino)-N-{1-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-5-carboxamide
N-{2-[(1-ethyl-3-methylpiperidin-3-yl)formamido]ethyl}-4-fluorobenzamide
2-(dimethylamino)-2-(3-methylphenyl)-1-[3-(pyridin-2-yl)azetidin-1-yl]ethan-1-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-1-ethyl-5-oxopyrrolidine-3-carboxamide
(2S,4S)-1-acetyl-4-[3-(dimethylamino)benzamido]-N,N-diethylpyrrolidine-2-carboxamide
N-[(3S,4R)-1-(1-benzothiophene-5-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
2-(1,2-oxazol-5-yl)-4-{pyrazolo[1,5-a]pyridin-7-yl}phenol
5-(dimethylamino)-2-[(3-phenyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
2-{4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperazin-1-yl}acetamide
1-ethyl-3,5-dimethyl-4-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-pyrazole
methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
6-(1-methyl-1H-imidazol-2-yl)-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyridazin-3-amine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridin-2-one
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-amino-4-(3-chloro-5-fluoro-4-methoxyphenyl)-6-ethyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-methyl-4-{[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}thiophene-2-carboxamide
(3R,4R)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
8-methyl-3-{[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-[2-(3-fluorophenyl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-[(1R,5R)-6-[(3-chloro-2,4-difluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
7-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-methyl-2,7-diazaspiro[4.5]decane
2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylacetamide
(4aS,8aR)-1-butyl-6-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridin-2-one
(2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(1-phenylethyl)-4H-1,2,4-triazole
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3,4-dihydropteridin-4-one
3-methyl-1-(4-{5-[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}phenyl)-1H-pyrazol-5-amine
2-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
(4aR,7aS)-1-(2-methylpropanoyl)-4-(quinolin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-(pyrazin-2-ylmethyl)-1H-indole-6-carboxamide
N-[2-(dimethylamino)ethyl]-1,3-dimethyl-N-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-(2,6-dimethylphenoxymethyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
6-{[(5-methylpyrazin-2-yl)methyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
4-(hydroxymethyl)-1-[3-(2-methoxyphenyl)benzoyl]azepan-4-ol
2-(1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
[4-(6-methoxypyridin-2-yl)phenyl]methanamine
2-(2H-1,3-benzodioxol-5-yloxy)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(2-methyl-1H-1,3-benzodiazol-1-yl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
N-(3-chloro-4-propanamidophenyl)-3-(1H-pyrazol-4-yl)benzamide
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-1,3-benzodiazole-5-carboxamide
N-(2-{[(2-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]amino}ethyl)acetamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
(3S,4S)-1-(2-ethoxypyridine-3-carbonyl)piperidine-3,4-diol