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N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)benzamide
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-{2-oxo-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethyl}-1λ6-thiolane-1,1-dione
2,6,8-trimethyl-N-[2-(1,3-thiazol-4-yl)ethyl]quinoline-4-carboxamide
N-[4-(4-{[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]amino}piperidin-1-yl)phenyl]benzenesulfonamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]acetamide
2-[4-(1,2-dihydroacenaphthylen-5-yl)-1H-pyrazol-1-yl]-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
2-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-(cyclopropylamino)-N-[3-(dimethylamino)-1-phenylpropyl]acetamide
(5S)-5-{[({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)(pyridin-2-ylmethyl)amino]methyl}pyrrolidin-2-one
5-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
9-(3-chloropyridin-2-yl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
8-{[4-(3-ethylpiperazine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
N-(2,2-difluoroethyl)-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
ethyl 1-{[4-(2-hydroxyethoxy)phenyl]methyl}-3-(2-phenoxyethyl)piperidine-3-carboxylate
6-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-9H-purin-2-amine
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)methylamine
2-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzoic acid
3-(2-hydroxyphenyl)-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-1H-pyrazole-5-carboxamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-3-propanamidobenzamide
N-benzyl-5-{[4-(oxan-4-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
N-cyclopropyl-3-[1-(4-ethyl-5-methylpyrimidin-2-yl)piperidin-4-yl]propanamide
(2S,4R)-4-(dimethylamino)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxylic acid
3-[2-(4-methoxyphenyl)ethyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
N-cyclopentyl-1-{1-[2-(4-methoxyphenoxy)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-(2,5-dimethoxyphenyl)-5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-5-methoxybenzamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
5-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1-(2-phenylethyl)piperidin-4-amine
6-methyl-N-[(4-sulfamoylphenyl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(5-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
5-methanesulfonyl-2-(piperidin-1-yl)-4-(piperidin-3-yl)pyrimidine
2,2-dimethyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)propanamide
N1,N3-dimethyl-5-[2-(thiophen-3-yl)-1H-imidazol-1-yl]benzene-1,3-dicarboxamide
2-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-4-(pyridin-2-yl)pyrimidine
6-cyclopropyl-N-{2-[ethyl(methyl)amino]butyl}pyrimidin-4-amine
1-(5-carbamoylpyridin-2-yl)-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid
N-{3-[(pyridin-3-yl)amino]propyl}-1H-pyrazole-4-carboxamide
6-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
[1-(5-{[(3-fluorophenyl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-(1H-1,2,4-triazol-1-yl)propan-1-one
8-[4-(4-fluorophenyl)oxane-4-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-(3,3-diphenylpiperidin-1-yl)ethan-1-one
(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-3-(prop-2-en-1-yl)piperidin-3-yl)methanol