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4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[(2-methylpyridin-4-yl)methyl]pyrimidin-2-amine
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperidine
3-chloro-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
6-[3,5-bis(trifluoromethyl)phenyl]-9H-purin-2-amine
1-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
5-(oxane-4-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-({[(3R,4R)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(1-carbamoylcyclopentyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-5-methylpyrimidine
2-(1-{[2-(1H-imidazol-2-yl)phenyl]methyl}pyrrolidin-2-yl)-1,3-thiazole
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]but-2-yn-1-one
3-benzyl-1-(2-phenylethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(2,3-dimethoxyphenyl)-9-methoxy-4-{[3-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 3-acetamido-1-[2-(1H-indol-3-yl)ethyl]-5-[(thiophen-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
7-[(3-methylphenyl)methyl]-2-(propan-2-yl)-2,7-diazaspiro[4.5]decane
2-(5-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidin-2-yl}-1-cyclohexyl-1H-1,2,4-triazol-3-yl)acetamide
5-(hydroxymethyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]furan-2-carboxamide
N-benzyl-2-(furan-2-yl)pyrrolidine-1-sulfonamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
5-(1-butanoylpyrrolidin-2-yl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}thiophene-2-carboxamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(2-fluorophenyl)ethan-1-one
3-{[(2-aminopyrimidin-4-yl)amino]methyl}-6-cyclopentyl-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
ethyl 2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)-1,3-oxazole-4-carboxylate
2-(2,4-dichlorophenoxy)-N-[(dimethyl-1,3-thiazol-5-yl)methyl]acetamide
1-(5-fluoro-1H-indole-2-carbonyl)-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(pyrrolidin-1-yl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
4-(4-methylphenoxy)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
(3S,4R)-4-(2-methoxyphenyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(2,5-dimethoxyphenyl)-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
N,3,5-trimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole-2-carboxamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-methyl-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-[(2-methylpyridin-4-yl)methyl]urea
2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
1-(4-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}phenyl)ethan-1-one
7-[4-(4-methoxyphenyl)butanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-(4-chlorophenyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}butanamide
4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-N-(2-methylphenyl)piperidine-1-carboxamide
2-methyl-7-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2,7-diazaspiro[4.5]decane
2,4-dimethyl-6-[1-(1-methylpiperidin-4-yl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyrimidine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2,5-dimethoxyphenyl)methyl]methylamine
N-(cyclohex-1-en-1-ylmethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-methoxy-N,3-dimethylbenzamide
9-[(3-fluoro-5-methylphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(3,4-difluorophenyl)methyl]-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide