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2-[3-(4-methoxypiperidine-1-carbonyl)benzenesulfonamido]-N,N-dimethylacetamide
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
2-{4-[3-(pyridin-2-yl)azetidine-1-carbonyl]piperidin-1-yl}acetamide
3-(6-methoxynaphthalene-2-carbonyl)-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine
2-(azepan-1-yl)-N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2,6,8-trimethylquinoline-4-carboxamide
3-(3-fluorophenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzamide
4-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
2-(3-chlorophenyl)-1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
N-methyl-4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]pyridin-2-amine
N-[2-(4-fluorophenyl)ethyl]-2-(1H-imidazol-2-yl)benzamide
(2S,4R)-4-[4-(3-cyanobenzenesulfonamidomethyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
4-methyl-1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroquinolin-2-one
3-(1-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-imidazol-2-yl)phenol
3-(4-methyl-1,3-thiazol-5-yl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}propanamide
6-(benzyloxy)-1-cyclohexyl-4-(1-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-2-one
4-(2-{[3-(azepane-1-carbonyl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethyl)benzene-1-sulfonamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclobutanecarboxamide
2-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidin-2-yl)pyridine
methyl 5-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
4-hydroxy-2-(thiophen-2-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]pyrimidine-5-carboxamide
8-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(4-fluoro-3-methylphenyl)-1-methyl-6-[(2-methyl-1H-imidazol-4-yl)methyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(1S,5R)-6-(cyclopropylmethyl)-3-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-hydroxy-2-methylpropan-2-yl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
5-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-(3-methoxyphenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
2-[2-(4-ethylpiperazin-1-yl)acetyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(1-benzyl-1H-pyrazol-4-yl)phenyl]acetamide
1-(2-fluorophenyl)-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}cyclopropane-1-carboxamide
4-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-yl}thiomorpholine
(3E)-1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pent-3-en-1-one
(1S,6R)-9-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
3-(1H-1,3-benzodiazol-2-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]propan-1-one
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
3-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-1H-indazole
cyclopentyl 4-[(2S)-2-amino-3-(1,3-thiazol-4-yl)propanamido]benzoate
N-methyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-{4-[(5-methylfuran-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-cyclopropanecarbonyl-N-(5-ethyl-1,3,4-oxadiazol-2-yl)piperidin-3-amine
4-(cyclopropylmethyl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine
6-(3-hydroxypiperidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
2-acetyl-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide
2-{5-[1-(2-fluorophenyl)-2,2-dimethylcyclopropyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-{[2-(benzyloxy)phenyl]methyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide