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2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-1-(morpholin-4-yl)ethan-1-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
9-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
8-(5-ethenylpyridin-2-yl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-2-[(4-fluorophenyl)methyl]morpholine
4-{3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}-1,5-dimethyl-1H-pyrazole
N,N-dimethyl-2-{[(2S)-2-(methylamino)hexanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-[(3-benzoylpiperidin-1-yl)methyl]-1,5-dimethyl-1H-pyrrole-2-carbonitrile
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-(1H-pyrazol-1-yl)butanamide
4-[(3aS,6aS)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-b]pyrrole-1-carbonyl]morpholine
3-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-[4-(1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-imidazol-2-yl)phenyl]acetamide
N-ethyl-2-(2-propyl-1H-1,3-benzodiazol-1-yl)-N-(pyridin-4-ylmethyl)propanamide
N-benzyl-2-ethyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrimidine-5-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]ethan-1-one
6-methyl-2-({2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}amino)-3,4-dihydropyrimidin-4-one
2-methoxy-5-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)phenol
2-[(2-fluorophenyl)methyl]-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,3-benzoxazole-6-carboxamide
1-cyclopentyl-4-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]pyrrolidin-2-one
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylsulfanyl)ethan-1-one
1-[3-(cyclopentyloxy)phenyl]-3-[2-(dimethylsulfamoyl)ethyl]urea
N-methyl-N-(2-phenylethyl)-1-(1,3-thiazol-2-ylmethyl)piperidin-3-amine
2-tert-butyl-4-hydroxy-N-[2-(2-oxoimidazolidin-1-yl)ethyl]pyrimidine-5-carboxamide
N-cyclopropyl-4-methoxy-2-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)oxy]benzamide
N-ethyl-2,6-dimethoxy-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyridine-3-carboxamide
2-[(2-methylpyridin-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(ethylamino)-4-methyl-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-thiazole-5-carboxamide
N-[2-(1H-pyrazol-1-yl)ethyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
3-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
3-phenyl-5-[3-(propan-2-yloxy)benzoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(2-ethoxyethyl)-N-[(4-methylpyridin-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3R,5S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,5-dimethyl-1H-pyrazole-3-carboxamide
1-cyclohexanecarbonyl-4-(cyclopropylmethyl)-1,4-diazepan-5-one
2-(2-oxo-1,3-oxazolidin-3-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
4-(3-chlorobenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-{[(1-methyl-1H-imidazol-2-yl)methyl](pyridin-4-ylmethyl)amino}ethan-1-ol
2-(2,3-dimethylphenoxy)-2-methyl-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propan-1-one
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
[4-(5-chloro-3-phenyl-1H-indole-2-carbonyl)morpholin-2-yl]methanamine
N,N-dimethyl-7-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(2-phenylpropyl)piperidine
3-(1H-indazol-4-yl)-1-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]urea
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(2S,4S)-4-amino-1-(3-methanesulfonylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methylpyridin-2-amine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2-fluorophenyl)methyl]methylamine
(2S,4R)-4-amino-1-hexanoyl-N-(propan-2-yl)pyrrolidine-2-carboxamide