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N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
2-(carbamoylamino)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
4-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
N-[(2-fluorophenyl)methyl]-N-propylcyclohex-3-ene-1-carboxamide
3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridin-2-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
7-(cyclohexylmethyl)-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[3-(2-chlorophenoxy)propyl]-5-cyclopropyl-N-methyl-1,3,4-oxadiazol-2-amine
1-(furan-2-ylmethyl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-3-carboxamide
(3R)-1-({3-ethoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)pyrrolidin-3-ol
(1R,3S)-7-[5-(4-chlorophenyl)-4-methyl-1H-pyrazole-3-carbonyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
(1S,6R)-3-[(3,5-dichloropyridin-4-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
2-{[4-(2-methoxy-5-methylphenyl)-5-(oxan-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(3R,4S)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-phenylpyrrolidin-3-amine
N-ethyl-3-[4-(morpholine-4-sulfonyl)phenyl]benzamide
2,4-dichloro-3-[(2,2-dimethylmorpholin-4-yl)methyl]phenol
3-methyl-8-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(dimethylamino)ethyl]-N-{[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}oxolane-2-carboxamide
methyl({[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl})[(3-methylthiophen-2-yl)methyl]amine
8-fluoro-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylquinoline-2-carboxamide
2-{benzyl[2-(dimethylamino)ethyl]amino}-2-(5-fluoro-2-methoxyphenyl)acetic acid
2-(3-fluoro-4-methoxyphenyl)-2-{methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amino}acetic acid
6-methyl-5-{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3-hydroxypiperidin-1-yl)-1-[4-(4-methoxyphenoxy)piperidin-1-yl]ethan-1-one
3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]-1-[1-(1H-1,2,4-triazol-5-yl)ethyl]urea
(4aR,7aS)-1-(2-methylpropyl)-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-5-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-(methylamino)-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-4-carboxamide
(3aS,7aR)-5-methyl-2-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}quinoline-3-carboxamide
ethyl 2-{4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl}acetate
N-[3-(oxolan-3-yl)propyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-amino-1-[(3,5-difluoro-4-methoxyphenyl)methyl]pyrrolidine-3-carboxylic acid
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(propylcarbamoyl)pyrrolidine-3-carboxylic acid
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl]propanoate
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
4-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
methyl N-{4-[5-(cyclopropylcarbamoyl)thiophen-2-yl]phenyl}carbamate
1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}butan-1-one
2-[4-(dimethylamino)phenyl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-5-[1-(2-methylpropyl)pyrrolidin-2-yl]thiophene-2-carboxamide
methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}){[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
8-(2-oxoimidazolidine-4-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-(2-phenoxyethyl)-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazine
3-(5-methylfuran-2-yl)-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
4-(furan-2-carbonyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-1,4-diazepane-1-carboxamide
4-(difluoromethoxy)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide