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N-(1-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
7-(propan-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-ethyl-3-{1-[2-(1H-pyrazol-1-yl)butanoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1,4-oxazepan-6-yl}methanol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(pyrazin-2-ylmethyl)acetamide
(3S,4R)-1-(3,4-difluorobenzoyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-(2-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-(pentan-3-yl)-1,2-oxazole-3-carboxamide
6-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2,3-dimethylquinoxaline
3-(4-methyl-1H-pyrazol-1-yl)-N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidine-2,5-dione
N-cyclopropyl-2-{[1-(3,3-dimethylcyclohexyl)piperidin-4-yl]oxy}-4-methoxybenzamide
2-methyl-8-{[3-(2-methylphenyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine
3-[2-(4-fluorophenyl)ethyl]-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
3-(2-methylpropyl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1,2-oxazole-5-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-hydroxyethyl)-5-methoxy-N-methylbenzamide
4-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1λ6-thiane-1,1-dione
(4aR,8aS)-1-(cyclohexylmethyl)-6-[(2-hydroxy-4-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-ethyl-5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}pyrimidin-2-amine
N,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(4-methylpyridin-2-yl)propan-2-yl]quinoline-4-carboxamide
N-[2-(5-methyl-4-{[3-(thiophen-2-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
3-(1H-imidazol-4-ylmethyl)-4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperazin-2-one
(1S,4S)-2-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(5-methyl-1H-pyrazol-1-yl)acetamide
5-{4-[(2-hydroxyethyl)amino]quinazolin-6-yl}-1,2-dihydropyridin-2-one
4-ethyl-1-methyl-3-{[1-(4-methylpyridine-3-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-[4-({4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-ol
3-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
1-(2,2-dimethylpropanoyl)-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(morpholine-4-sulfonyl)benzoic acid
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
6-[3-(4-methylpiperazin-1-yl)pyrrolidine-1-carbonyl]quinoline
1-[4-(hydroxymethyl)benzoyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-tert-butyl-2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoacetamide
5-methyl-5-{1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]piperidin-4-yl}imidazolidine-2,4-dione
3-[5-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)thiophen-3-yl]prop-2-yn-1-ol
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-(3-methanesulfonylpropanoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-(cyclobutylmethyl)-3-(3-methoxyphenyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
ethyl 3-({8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}amino)propanoate
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
3-{[1-(4-aminopyridine-2-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-ethyl-5-({3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
2-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
1-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea