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1-{[4-(2-methylphenyl)phenyl]methyl}piperidine-3-carbonitrile
5-(3-methylphenyl)-2-(pyridin-4-yl)-4-[1-(thiophen-2-ylmethyl)piperidin-4-yl]pyrimidine
(3S,4S)-1-(1-benzofuran-5-ylmethyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1-(4-fluorophenyl)-4-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]butane-1,4-dione
(4aS,8aR)-1-(4-hydroxybutyl)-6-[3-(1,2-oxazolidin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
3-(2,2-dimethyloxan-4-yl)-3-ethyl-1-[3-(pyridin-3-yl)phenyl]urea
N4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N4-methyl-5,6,7,8-tetrahydroquinazoline-2,4-diamine
{3-[5-(2-methylfuran-3-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
2-(1-ethyl-3-oxopiperazin-2-yl)-N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}acetamide
4-acetyl-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)benzamide
N-(2-hydroxybutyl)-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2-propylpyridine-4-carboxamide
3-{1-[2-(piperidin-1-yl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(5-methylthiophen-2-yl)methyl]piperidin-4-ol
(3S)-3-({[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}amino)azepan-2-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-cyclopropyl-4-methoxy-2-({1-[1-(4-methylphenyl)propan-2-yl]piperidin-4-yl}oxy)benzamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
(1R,3S)-N-benzyl-1-hydroxy-3-methoxy-N-methyl-7-azaspiro[3.5]nonane-7-sulfonamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(2-chloro-6-fluorophenyl)ethan-1-one
1-(1-cyclopentylpiperidine-3-carbonyl)-4-(1,3-thiazol-2-yl)piperazine
1-(4,6-dimethylpyrimidin-2-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}piperidin-4-amine
3-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
1-[2-(benzyloxy)acetyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-phenyl-N-{1-[1-(4,4,4-trifluorobutan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
4-(azepane-1-carbonyl)-8-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
(1S,9aR)-1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-octahydro-1H-quinolizine
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]acetamide
(3aR,6aS)-5-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
1-(4-chlorophenyl)-4-(2,5-dimethylfuran-3-carbonyl)-5-methylpiperazin-2-one
(1R,3S,5S)-8-({5-[(5-propylfuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-8-azabicyclo[3.2.1]octan-3-ol
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[3-(5-methylfuran-2-yl)butyl]amine
9-(2-methoxyethyl)-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-amino-4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-(3-phenyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-amino-6-(2,2-dimethyloxan-4-yl)-4-(4-hydroxy-3-methoxyphenyl)-5-methylpyridine-3-carbonitrile
5-chloro-7-methoxy-N-[3-(methylamino)propyl]-1-benzofuran-2-carboxamide
1-(3-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)azepan-2-one
7-({[2-(1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)-5-(2-chloroprop-2-en-1-yl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-fluorophenyl)methyl]-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
4-ethyl-N-[1-(methoxymethyl)cyclopentyl]-2-methyl-1,3-thiazole-5-carboxamide
1-(benzenesulfonyl)-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
N-(3-methyl-1-propyl-1H-pyrazol-5-yl)-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
4-benzyl-3-[1-(1H-imidazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pentan-3-yl)acetamide
1-(carbamoylmethyl)-N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]piperidine-3-carboxamide
4-(4-methoxyphenyl)-2-methyl-1-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
N-(2,2,2-trifluoroethyl)-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide