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2-(1-ethylpiperidin-4-yl)-1-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
5-(4-ethylpiperazin-1-yl)-N-[(2-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]urea
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-cyclopentyl-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
{3-[2-(1-benzoylpiperidin-3-yl)-1H-imidazol-1-yl]propyl}dimethylamine
7-(cyclopropylmethyl)-2-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
1-(cyclohexylmethyl)-N-methyl-5-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
4-(1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)morpholine
(2R)-1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
2,7,8-trimethyl-N-[1-(pyrimidin-4-yl)ethyl]quinoline-4-carboxamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(1-propylpiperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[4-fluoro-3-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]acetic acid
1-[4-(hexylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[2-methoxy-5-(morpholin-4-ylmethyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[1-(dimethoxy-1,3,5-triazin-2-yl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(4-benzylpiperazin-1-yl)-3-[1-(4-methoxybenzoyl)piperidin-3-yl]propan-1-one
3-{2-[(3-hydroxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
N-ethyl-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]-N-phenylbenzamide
(1R,5R)-6-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
8-(5-fluoro-2-methoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[4-(thiomorpholine-4-sulfonyl)benzoyl]azepane
7-(2-hydroxyethyl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-dihydroquinoxalin-2-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})(3,3,3-trifluoro-2-methylpropyl)amine
(3aR,6aR)-2-cyclopropanecarbonyl-5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[4-(propan-2-yl)phenyl]-1-(3,4,5-trimethoxybenzoyl)piperidin-3-amine
5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{2-[(3S,4S)-4-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-methanesulfonyl-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
3-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]but-2-ynamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-1H-imidazole-2-carboxamide
5-(dimethylamino)-2-{2-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
(2S,4S)-4-amino-1-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-[(3-fluorophenyl)methyl]-9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2R,6R)-11-methoxy-4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-cyclopentyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
2-(morpholin-4-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-1-carboxamide
1-(5-methyl-2-phenylfuran-3-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(2-phenylpropyl)acetamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
8-[(4-acetylphenyl)carbamoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-{5-[3-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)propyl]-1,2,4-oxadiazol-3-yl}pyridine
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}propanamide