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(2S,4S)-N-ethyl-1-methyl-4-[4-(4-methylpiperazin-1-yl)benzamido]pyrrolidine-2-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
(2S,4R)-4-amino-N-methyl-1-(4-phenylbenzenesulfonyl)pyrrolidine-2-carboxamide
7-(2-cyclohexylethyl)-2-(2-hydroxy-4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
3,4,7-trimethyl-N-({5-methyl-2-[2-(oxolane-2-amido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-indole-2-carboxamide
5-methyl-1-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
(1-{[methyl({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}cyclopropyl)methanol
1-{4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(benzyloxy)ethan-1-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[(3S,4R)-1-(2-methoxypyridine-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
1-(3-methyl-1,2,4-thiadiazol-5-yl)-3-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]urea
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]pyrazine-2-carboxamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-methyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(dimethylamino)-2-(4-methylphenyl)-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]acetamide
4-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}-1,4-oxazepan-5-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methyl-1,3-thiazole-5-carboxamide
1-(6-hydroxy-4-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
6-methyl-2-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}-4-(thiomorpholin-4-yl)quinazoline
N-[2-(ethanesulfonyl)ethyl]-5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-amine
2-(2,4-difluorophenoxy)-1-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethan-1-one
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
[(2S,6S)-4-[2-(benzyloxy)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]propanamide
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-2-fluoro-5-sulfamoylbenzamide
(2S)-N-[3-(3-chlorophenyl)phenyl]-1-methylpyrrolidine-2-carboxamide
(1R,2S,4R)-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-[4-(1-methoxyethyl)phenyl]pyridin-3-amine
1-{2-[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-({5-[1-(3,3-dimethylbutyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-[(3R,4S)-1-[(2,6-dioxo-1,2,3,6-tetrahydropyrimidin-4-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-(piperidin-1-yl)piperidine
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azepane
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazole-5-carboxamide
2-(4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazin-1-yl)-1-(piperidin-1-yl)ethan-1-one
3-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]sulfamoyl}-N-[2-(methylamino)ethyl]benzamide
N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
4-fluoro-N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}benzamide
N-{[3-methyl-7-(2-phenylpropanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[2-(pyrazin-2-yl)ethyl]acetamide
4-(3-chloro-4-methoxyphenyl)-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-5-methyl-1,2-oxazole-3-carboxamide
4-(3-{6-[(dimethylamino)methyl]-1,4-oxazepane-4-carbonyl}phenyl)-2-methylbutan-2-ol
ethyl(oxan-4-ylmethyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
3-{2-[2-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
2-[4-(butane-1-sulfonyl)morpholin-3-yl]-N-(pyridin-4-ylmethyl)acetamide
4-[1-(1-cyclopentylpiperidin-4-yl)piperidine-3-carbonyl]morpholine
6-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
5-(3,6-dimethyl-1-benzofuran-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole