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1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxy-2-(4-methoxyphenyl)ethan-1-one
N-[1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)pyrrolidin-3-yl]acetamide
(1S,5R)-3-cyclobutanecarbonyl-6-phenylmethanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
6-(1,4-oxazepan-4-ylmethyl)-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
methyl 4-{[5-(4-chlorophenyl)-1,2,4-triazin-3-yl]amino}butanoate
4-({3-[(2,5-dimethylphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-2-one
3-[1-(1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)piperidin-3-yl]benzoic acid
1-(4-methoxyphenyl)-3-methyl-5-{[1,2,4]triazolo[1,5-a]pyrimidin-6-ylmethyl}-1H-1,2,4-triazole
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
1-{1-[6-(4-ethyl-1,4-diazepan-1-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
3-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(4-chlorophenyl)(phenyl)methyl]-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-(2-phenoxyethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(1H-1,3-benzodiazol-1-yl)-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}propanamide
3-(1-{[4-(benzyloxy)phenyl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
N-tert-butyl-2-({4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-6-yl}amino)acetamide
3-{3-[1-(but-3-en-1-yl)-1H-pyrazol-3-yl]phenyl}-6-methoxypyridazine
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}acetamide
2-[(3-{[1-(2,4-dimethoxyphenyl)ethyl](methyl)carbamoyl}phenyl)amino]acetic acid
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,3-thiazole-4-carboxamide
1-(3-cyano-2-methoxypyridin-4-yl)-4-hydroxypiperidine-4-carboxylic acid
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole
1-(4-fluorophenyl)-2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethan-1-ol
N-(furan-3-ylmethyl)-N-methyl-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
2-methoxy-N-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
5-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole
{3-[(3-chlorophenyl)methyl]-1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-3-yl}methanol
1-ethyl-4-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-1H-pyrrole-2-carbonitrile
1-[(3-methylphenyl)methyl]-4-[2-(pyrrolidin-1-yl)acetyl]piperazin-2-one
(1s,4s)-4-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}cyclohexan-1-ol
1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
1-[2-(dimethylamino)-6-(6-methylpyridazin-3-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
6-[(furan-2-ylmethyl)amino]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-(2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)methanesulfonamide
2-(6-methylpyridine-2-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
2-cyclohexyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(4-fluorophenyl)acetamide
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-phenyl-1,3-thiazole-2-carboxamide
6-(1-methylpiperidin-3-yl)-2-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperazine-1-sulfonamide
3-(azepane-1-carbonyl)-6-methyl-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-4-one
methyl({[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-[(3R,4S)-4-(dimethylamino)-1-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]piperidin-3-yl]propanoic acid
2-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
ethyl 1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate