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N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-2-hydroxy-N-(2-methoxyethyl)acetamide
6-[4-(piperidine-1-sulfonyl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]quinoxaline-6-carboxamide
N-[2-(3-ethoxyphenoxy)ethyl]-N-methyl-2-(2-oxo-1,2-dihydroquinolin-1-yl)acetamide
1-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-[(1-benzyl-1H-imidazol-5-yl)methyl]imidazolidin-2-one
3-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-1-(pyridin-3-ylmethyl)-1-(thiophen-3-ylmethyl)urea
5-acetyl-N-methyl-N-(quinolin-5-ylmethyl)thiophene-2-carboxamide
2-benzyl-8-(pyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-amino-1-[(2,6-dichloro-3-hydroxyphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
ethyl 1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
7-(piperidin-3-yl)-N-[2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(4-phenyl-1H-pyrazol-5-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
methyl 2-{2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methylacetamido}acetate
1-{4-[4-({5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}amino)piperidin-1-yl]phenyl}pyrrolidin-2-one
N-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]acetamide
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
3-(3-fluorophenyl)-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
1-{2-hydroxy-3-[3-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
2-[5-(oxolan-2-yl)thiophene-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-(1H-imidazol-4-ylmethyl)-4-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-1,4-diazepane-6-carboxylic acid
5-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-1H-indazol-3-amine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-{[(3-chloro-4-methylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[2-(benzyloxy)ethyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
7-(3-chlorophenyl)-4-(2-methyloxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-azaspiro[5.5]undecan-9-amine
{3-[(3-chlorophenyl)methyl]-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl}methanol
methyl 5-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1R,7S)-3-(2-ethoxyethyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4,6-dimethyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
(2S,4S)-N-methyl-4-[4-(2-{[(2-methylphenyl)carbamoyl]amino}propan-2-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
1-({[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]carbamoyl}methyl)piperidine-4-carboxamide
1-cyclopentyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
4-(4-chlorophenyl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}butan-1-one
2-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2,2-dimethyl-N-(1-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-5-phenylpentanamide
7-(2-hydroxyethyl)-2-(pent-2-yn-1-yl)-2,7-diazaspiro[4.5]decan-6-one
5-chloro-N-methyl-N-(1,2-oxazol-5-ylmethyl)-3-phenyl-1H-indole-2-carboxamide
1-{[(5-fluoro-2-methylphenyl)carbamoyl]methyl}-5-oxopyrrolidine-3-carboxylic acid
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-{3,5-dimethyl-4-[(E)-2-phenylethenyl]-1H-pyrazol-1-yl}acetamide
N-[2-(4-methylpiperazin-1-yl)butyl]-6-(piperidin-1-yl)pyrimidin-4-amine
4-{[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]methyl}-1-[(2R)-pyrrolidin-2-ylmethyl]piperidine
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
1-[1-(morpholine-2-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one