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8-{[3-(4-benzylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}quinoline
[(2S)-1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-2-yl]methanol
6-[(diethylamino)methyl]-N-(1,3-dihydro-2-benzofuran-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-(2-methoxyethyl)-8-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3S,4R)-4-propyl-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl]methanesulfonamide
ethyl 1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}piperidine-3-carboxylate
7-(2-methoxyethyl)-2-(4-methylpiperazine-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[cyclohexyl(methyl)amino]-3-(3-{[methyl(prop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]propan-1-one
5-(2-fluorophenoxymethyl)-N-[(3-hydroxyphenyl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-ol
(3R,7S,8aS)-7-{[(4-chlorophenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-methyl-6-(3-methylpiperidine-1-carbonyl)-N-[2-(morpholin-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
N,N-dimethyl-2-[(1S,5R)-6-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-(1-benzofuran-2-carbonyl)-6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
1-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
N-methyl-N-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}cyclopentanamine
(1R,5R)-6-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
{1-[1-(2-phenyl-1H-imidazole-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-N-(6-methylpyridazin-3-yl)benzamide
2-(2-benzyl-1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
N-[(3-chlorophenyl)methyl]-2-ethyl-N-propylpyrimidine-5-carboxamide
N-[2-(2-chlorophenoxy)ethyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
1-benzyl-5-[(diethylcarbamoyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-cyclopentyl-N,1-dimethyl-N-[(3-methyloxetan-3-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}thiomorpholine
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-methoxypyridine-3-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrazole-3-carboxamide
[9-(pyridin-3-ylmethyl)-3-(thiophen-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
6-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyrimidin-4-amine
3-[1-(2-hydroxyethyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]-1-phenylpropan-1-one
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-methylthieno[2,3-d]pyrimidin-4-amine
1-(6-chloro-1,3-benzothiazol-2-yl)-N-(1H-pyrazol-3-ylmethyl)piperidin-4-amine
2-{1-[(3S,4R)-4-ethoxyoxolan-3-yl]-1H-imidazol-2-yl}benzoic acid
6-methoxy-4-[(4-methoxynaphthalen-1-yl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
4-(1-benzofuran-2-yl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-(oxan-2-ylmethyl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-[(3R,4S)-1-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
2-[4-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
1-(2H-1,3-benzodioxole-5-carbonyl)-4-[2-(naphthalen-1-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
N-[3-(3-ethylphenoxy)propyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N,N-dimethyl-4-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]aniline
6,6-dimethyl-N-[2-(3-methylthiophen-2-yl)ethyl]-5-oxothiomorpholine-3-carboxamide
2-methyl-4-[4-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)phenyl]butan-2-ol
8-(1H-indol-2-ylmethyl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({4-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)piperidine-4-carbonitrile
(3R,4R)-1-{[4-(furan-2-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol