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(3S,4S)-4-cyclopropyl-1-[3-(2-oxopiperidin-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
3-(4-chlorophenyl)-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-phenylpropanamide
6-[(diethylamino)methyl]-N-(5-methylpyridin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1-(thiomorpholin-4-yl)propan-1-one
1-[benzyl(methyl)amino]-3-[4-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
5-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
1-{4-[(3S)-3-hydroxypyrrolidin-1-yl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-[(1S,2S)-2-hydroxycyclohexyl]-3-(5-methyl-2,1,3-benzothiadiazol-4-yl)urea
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2-(pyrrolidin-3-yl)benzamide
1-(5-ethylthiophene-3-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-({3-[(dimethylamino)methyl]phenyl}methyl)-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
5,7-dimethyl-N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}pyrido[2,3-d]pyrimidin-4-amine
N-[2-(dimethylamino)ethyl]-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
ethyl 4-{2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetyl}piperazine-1-carboxylate
7-(6-aminopyridine-3-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(2-methoxyphenyl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
1-[1-(3-fluorophenyl)-3-[hydroxy(phenyl)methyl]-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N-({5-[(3-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
3-benzyl-4-[1-(2-methoxyacetyl)piperidine-4-carbonyl]piperazin-2-one
1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-5-[1-(1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
1-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
4-[5-(1H-imidazol-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
5-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
1-(adamantan-2-yl)-N-(2H-1,3-benzodioxol-5-yl)piperidin-3-amine
(3aS,6aS)-2-acetyl-5-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[4-(2-phenylphenyl)pyridin-2-yl]methanol
dimethyl(1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]phenyl}ethyl)amine
dimethyl({2-[4-(5-methyl-1H-pyrazole-3-carbonyl)morpholin-2-yl]ethyl})amine
N-(2,3-dichlorophenyl)-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
8-(1-methylcyclopropanecarbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N,3-diethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-hydroxyadamantane-1-carboxamide
4-benzyl-3-ethyl-1-[2-(pyridin-3-yloxy)acetyl]-1,4-diazepan-5-one
methyl 3-benzamido-5-[(oxan-4-yl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5,7-dimethyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
N-[2-(1H-imidazol-4-yl)ethyl]-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
N-methyl-N-[3-(2-methylphenoxy)propyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
2-{[5-cyclopropyl-4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-methylpyrido[2,3-d]pyrimidin-4-amine
(3S,4S)-1-[(1-phenyl-1H-pyrazol-5-yl)methyl]-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyrrolidin-3-ol
5-(2,4-dimethoxyphenyl)pyridin-2-amine
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-2-ethyl-N-(2-methoxyethyl)butanamide
2-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}propan-2-ol
1-benzyl-N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}piperidin-4-amine
5-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate