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2-{[5-({[(2-ethoxyphenyl)methyl](ethyl)amino}methyl)pyrimidin-2-yl]amino}acetic acid
2-(4-{[(2-methoxyethyl)(1,3-thiazol-2-ylmethyl)amino]methyl}phenyl)-5,6-dimethyl-3,4-dihydropyrimidin-4-one
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
5-amino-4-chloro-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
1-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-yl]-4-phenylbutane-1,4-dione
2-(5-acetylthiophen-3-yl)-1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-3-sulfamoylthiophene-2-carboxamide
2-(dimethylamino)-8-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-ethyl-4-(2,3,6-trimethylquinoline-4-carbonyl)piperazin-2-one
1-[4-({[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]amino}methyl)phenyl]pyrrolidin-2-one
2-(oxolan-2-ylmethyl)-8-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
8-(1-benzothiophene-2-carbonyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
5-methanesulfonamido-N-methyl-1-(2-phenylethyl)-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N4,4-dimethyl-N1-[4-(3-methylphenyl)phenyl]piperidine-1,4-dicarboxamide
4-[(1R,5S)-3-azabicyclo[3.3.1]nonan-3-yl]-6-(propan-2-yl)pyrimidin-2-amine
4-(4-benzyl-1H-1,2,3-triazol-1-yl)-N-(2-methylphenyl)piperidine-1-carboxamide
dimethyl({[(3R,4S)-1-[(2E)-2-methylbut-2-en-1-yl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
methyl (1R,3S,3aR,6aS)-1-ethyl-3-(4-methanesulfonylphenyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(oxan-3-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
1-(1-{[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(4aS,7aR)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}acetamide
N3-cycloheptyl-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(1-phenylethyl)-3-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(cyclobutylamino)-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-methyl-4-(4-methylphenyl)piperazine
1-(5-{[3-(methoxymethyl)piperidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)-4-methyl-1,4-diazepane
8-[2-(3,4-dimethylphenoxy)ethyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
[5-({3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}methyl)furan-2-yl]methanol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,3,6-trimethyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
[(3R,4R)-1-(5-chloronaphthalene-1-carbonyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
2-[(2,2-dimethyloxan-4-yl)(methyl)amino]-N-[2-(4-methoxyphenyl)ethyl]acetamide
6-[(diethylamino)methyl]-N-(2,3-dihydro-1H-inden-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-(cyclopropylmethyl)-5-[4-(1H-imidazol-1-yl)benzoyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(2,4-dimethylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(ethylsulfanyl)ethyl]-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
1-methyl-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(3-{7-ethyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}propoxy)benzamide
2-butyl-4-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxopiperazine-1-carboxamide
3-[4-(dimethylamino)phenyl]-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-[1-(2,5-difluorophenyl)cyclopropyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
4-(4-{[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide