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3-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carbonyl]pyridin-2-ol
1,6-dimethyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
(1s,4s)-N-[(1-benzylpiperidin-4-yl)methyl]-4-hydroxy-N-methylcyclohexane-1-carboxamide
2-(4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
N-(1-cycloheptylpiperidin-3-yl)-3-phenylprop-2-ynamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
1'-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(3-chlorophenyl)-4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-(oxolane-2-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(morpholine-4-carbonyl)-N-(oxan-3-ylmethyl)benzene-1-sulfonamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-[4-(2,5-dimethylfuran-3-carbonyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile
3-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-2-ol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(pyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-({5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-1-ol
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2-oxoazepan-1-yl)acetamide
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperidine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}isoquinoline-1-carboxamide
1-(cyclohexylmethyl)-N3-[(1-methylpiperidin-3-yl)methyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(1,2-diphenylethyl)({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]furan-2-carboxamide
2-phenyl-N-[2-(pyridin-3-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
2-(3-methoxypropyl)-9-(1H-pyrazole-4-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
4-methyl-9-[3-(propan-2-yl)-1,2-oxazol-5-yl]-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
1-[(6-methoxy-2H-chromen-3-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-(furan-2-yl)-5-[1-(2-methoxypyridin-3-yl)-1H-imidazol-2-yl]pyrimidine
1-[3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
8-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
3-(3-hydroxy-3-methylbutyl)-N-(1-propylcyclopropyl)benzamide
5-methyl-4-{[2-(pyridin-3-yloxy)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
9-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
[4-({1-[(3,4,5-trimethoxyphenyl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
2,6,8-trimethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]quinoline-4-carboxamide
methyl 1-(2-methoxyethyl)-3-(3-methylbutanamido)-5-{[(4-methylphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[4-(methoxymethyl)benzoyl]-1,4-diazepane-6-carboxylic acid
methyl[3-(morpholin-4-yl)propyl]{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
(3S)-3-{[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}-3-phenylpropan-1-ol
2-(dimethylamino)-7-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{2-[ethyl(methyl)amino]-2-methylpropyl}-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-methylbut-2-en-1-one
3-{[(2-ethoxyethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
6-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}quinoline