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N-(2-{1-[benzyl(methyl)sulfamoyl]piperidin-2-yl}ethyl)acetamide
N-[3-(1,3-benzothiazol-2-yl)propyl]-1H-1,2,3-triazole-5-carboxamide
3,5-dimethyl-N-[3-(pyridin-4-yl)propyl]adamantane-1-carboxamide
(3aR,6aR)-N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-(4-fluorophenyl)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
3-[(3R,4S)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridazine
4-[5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
5-[(quinolin-8-yloxy)methyl]-N-(1H-1,2,4-triazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
4-(cyclopropylmethyl)-1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-{3-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
2-(4-chloro-1H-pyrazol-1-yl)-N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
(3R,7S,8aS)-7-{[(2,5-difluorophenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-methyl-2-(phenoxymethyl)-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-{5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
1-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
N-(4-chloro-2-methylphenyl)-3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carboxamide
(2R,4S)-4-hydroxy-1-[4-(propylamino)benzoyl]piperidine-2-carboxylic acid
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(morpholin-3-yl)acetamide
N-(2-hydroxyethyl)-3-(1-methyl-1H-pyrrol-2-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-5-carboxamide
N-[2-(4-chlorophenoxy)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(morpholin-4-yl)propan-1-one
2,5-dimethyl-N-[(1R,3S)-3-{methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}cyclopentyl]furan-3-carboxamide
4-(2,5-dimethylphenyl)-6-methoxypyrimidin-2-amine
2-[4-({3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
4-(4-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
(2S)-2-(3,3-diphenylpiperidine-1-carbonyl)pyrrolidine-1-carboxamide
(3S)-1-{[2-(4-fluorophenyl)phenyl]methyl}pyrrolidin-3-ol
methyl (2S)-1-[6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carbonyl]pyrrolidine-2-carboxylate
N-[(4-phenyloxan-4-yl)methyl]oxolane-3-carboxamide
N-tert-butyl-4-({[1-(ethoxymethyl)cyclopropyl]methyl}sulfamoyl)benzamide
(4aR,8aS)-6-[4-(piperidin-1-yl)benzoyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
[(4-ethylphenyl)methyl]({[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-phenyl-5-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2-oxazole
2-{[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
4-(3-hydroxy-3-methylbutyl)-N-[2-(1H-imidazol-1-yl)ethyl]benzamide
4-methyl-6-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-phenylpyrimidine
1-[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-methyl-3-(1-phenylmethanesulfonylpiperidin-3-yl)-N-[2-(pyridin-2-yl)ethyl]propanamide
5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
4-{1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperidin-3-yl}benzoic acid
3-(1H-1,2,3-benzotriazol-1-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
1-methanesulfonyl-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazine
(3R,4R)-4-amino-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-3-ol
(3S,5R)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide