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2-{2,7-diazaspiro[4.5]decan-2-ylmethyl}benzonitrile
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-N,N-dimethylacetamide
6-{methyl[(3-methylpyridin-2-yl)methyl]amino}-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
N-butyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
3-butyl-1-methyl-4-{2-[methyl(phenyl)amino]acetyl}piperazin-2-one
3-[2-(1-cyclopentylpiperidin-4-yl)ethyl]-7-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
8-(2-amino-9H-purin-6-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenoxypropanamide
2-amino-6-(propan-2-yl)-N-[(trimethyl-1H-imidazol-2-yl)methyl]pyrimidine-4-carboxamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
N-(5-chloro-2-methoxyphenyl)-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide
3-(4-methoxyphenyl)-N-methyl-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-2-(methoxymethyl)piperidine
2-(dimethylamino)-2-(4-fluorophenyl)-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]acetamide
3-(2-ethylbutyl)-8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-1-(propan-2-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
N-benzyl-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(2-chlorophenyl)acetamide
N-(4-fluorophenyl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-amine
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-[3-(azepan-1-yl)propyl]-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]pyridine-2-carbonitrile
5-acetyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]thiophene-3-carboxamide
3-(2,6-dimethylphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
N-(2-{1-[(2,6-dichloro-3-hydroxyphenyl)methyl]piperidin-2-yl}ethyl)acetamide
2-[1-(cyclohexylmethyl)-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-5-methyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
[2-ethoxy-5-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]methanol
2-[4-(adamantan-1-yl)piperazine-1-carbonyl]-5-methoxy-4H-pyran-4-one
2-(dimethylamino)-N-[2-(1H-imidazol-1-yl)ethyl]-6-phenylpyridine-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(1,3,7-trimethyl-1H-indol-2-yl)formamido]acetic acid
1-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidine-1-carbonyl]cyclopropane-1-carboxamide
3-benzyl-8-[(3-chloro-4-hydroxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
N,N-bis(furan-2-ylmethyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)pyridine
[(1-{[1-(1H-indole-6-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]dimethylamine
1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}azepane
2,4-dimethyl-N-[4-(4-{[3-(1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]benzamide
(2E)-N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]-3-phenylprop-2-enamide
ethyl 4-(2-phenoxyethyl)-1-propylpiperidine-4-carboxylate
1-[2-(3-cyclohexyl-1,2,4-oxadiazol-5-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,5-dimethyl-N-[2-(4-methylphenoxy)ethyl]-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(3-methoxyphenoxymethyl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
4-[2-(oxolan-3-yl)ethyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide