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1-acetyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
5-[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(1R,5S)-6-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-6-azabicyclo[3.2.1]octane
3-methyl-1-[4-(oxan-2-ylmethoxy)phenyl]-3-[(5-propyl-1H-pyrazol-3-yl)methyl]urea
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
2-[5-(methanesulfonylmethyl)pyridin-2-yl]-N,N-bis(propan-2-yl)benzamide
2-[(2-chlorophenyl)methyl]-4-(3-fluoro-2-methoxybenzoyl)morpholine
1-[(2-methoxyphenyl)methyl]-N-{2-[methyl(2-phenylethyl)amino]ethyl}-6-oxopiperidine-3-carboxamide
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperidine
6-chloro-2-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
4-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-1-(3-chlorophenyl)piperazin-2-one
3-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,3-thiazole-4-carboxamide
4-ethyl-1-methyl-3-{1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-methoxy-2-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]pyridine
3-(3-hydroxy-1,2-oxazol-5-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
1-(3-cyclopentylpropyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
2-(methylsulfanyl)-3-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyridine
5-[(2-chloro-4-fluorophenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-N-{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}benzamide
4-[(6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridin-3-yl)methyl]morpholine
2-(3-hydroxypiperidin-1-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
4-(4-{[(4,6-dimethylpyrimidin-2-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
N-(2-hydroxyethyl)-2-{[(3-methylphenyl)methyl]amino}-1-propyl-1H-1,3-benzodiazole-5-carboxamide
3-cyclopentyl-1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
2-(5-methyl-4-phenylthiophene-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
(2S,4S)-1-cyclohexyl-4-(4-ethenylbenzamido)-N-ethylpyrrolidine-2-carboxamide
4-phenyl-3-[1-(1-propylpiperidin-4-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N,2-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}thieno[3,2-d]pyrimidin-4-amine
9-[4-(oxolan-2-ylmethyl)piperazin-1-yl]-3-azaspiro[5.5]undecane
1-methyl-4-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]imidazolidin-2-one
methyl 3-[(3S,4R)-1-[(2-methylphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
2-{6-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
3-chloro-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)benzoic acid
1-(4-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}thiophen-2-yl)ethan-1-one
4-(2-methoxyphenoxy)-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-4-carboxylic acid
2-{4-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]phenoxy}ethan-1-ol
1-benzyl-3-(pyridin-2-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-2-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamido]-3-(4-hydroxyphenyl)propanoic acid
8-cyclohexyl-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}thiophene-2-sulfonamide
3-(2-chlorophenyl)-3-(2-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1-methylpyrrolidine-2,5-dione
1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
3-({1-[(4-carboxyphenyl)methyl]pyrrolidin-3-yl}methyl)benzoic acid
2-(3-chloropyridin-2-yl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane