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(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(3-fluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(furan-3-carbonyl)piperidin-4-yl]propanamide
N-cyclopentyl-3-[5-(1-ethylpiperidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
6-{3-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
2-[4-(1-ethoxyethyl)phenyl]-3-(piperidine-1-carbonyl)pyridine
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
4-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
4-(1H-imidazol-1-yl)-N-methyl-N-[1-(pyridin-3-yl)propyl]benzamide
6-(diethylamino)-1-(4,4,4-trifluorobutyl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
6-methoxy-4-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
N-[(3S,4R)-4-(propan-2-yl)-1-(1,3-thiazol-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-6-methylpyridin-2-amine
2-(dimethylamino)-2-(3-fluorophenyl)-1-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}ethan-1-one
2-(3-hydroxyphenyl)-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-methyl-4-(pyrrolidin-3-yl)-N-(quinolin-6-ylmethyl)benzamide
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,5-dihydro-1H-pyrrole
N,2-dimethyl-4-phenyl-N-[1-(pyridin-3-yl)propyl]pyrimidine-5-carboxamide
N-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)piperidin-3-amine
N-[3-(4-methylbenzenesulfonamido)propyl]-2-(morpholin-2-yl)acetamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-hydroxy-4-(methylsulfanyl)butan-1-one
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-methylpentane-1,2-dione
N-methyl-2-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)acetamide
1-[(4-fluorophenyl)methyl]-5-[1-(methoxymethyl)cyclopropanecarbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-(furan-3-ylmethyl)-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
[(1-cyclopentylpiperidin-4-yl)methyl][(4-methyl-4H-1,2,4-triazol-3-yl)methyl](oxolan-2-ylmethyl)amine
1-[4-(3-hydroxyphenyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
4-ethyl-3-({1-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)oxolane-2-carboxamide
(4S)-1-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-3,3,4-trimethylpiperidin-4-ol
6-ethoxy-3-{[4-(1-hydroxyethyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-{5-[1-(2-methoxy-2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]urea
5-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-1,2-dihydropyridin-2-one
2-{[1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}acetamide
(1S,5R)-6-(furan-2-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-2-(propylsulfanyl)pyrimidine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]propanamide
(2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]carbamoyl}pyrrolidine-2-carboxylic acid
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
14-(3-ethenylphenyl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[2-(1H-imidazol-2-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-({[(2-methylphenyl)methyl](prop-2-en-1-yl)amino}methyl)phenol
N-({4-[benzyl(ethyl)amino]quinazolin-2-yl}methyl)-2-(3-methoxyphenyl)acetamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(3-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenyl)ethan-1-one
6-(1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}piperidin-3-yl)pyrimidin-4-ol
5-benzyl-3-[2-(pyridin-2-yl)ethyl]-5-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione