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N-cyclohexyl-3-[2-(4-hydroxy-3,5-dimethylphenyl)-1H-imidazol-1-yl]propanamide
(cyclopropylmethyl)({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})propylamine
N5-[(5-ethylpyridin-2-yl)methyl]-N6-(3-methoxypropyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N,N-dimethyl-N'-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)butanediamide
2-(3,5-difluorophenyl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
4-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-(pyridin-4-yl)quinoline
4-(1-ethyl-1H-imidazol-2-yl)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
2-acetyl-8-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
5-amino-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-phenyl-1H-pyrazole-3-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
2-(benzylsulfanyl)-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}pyrimidine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(7-methyl-2-oxo-2H-chromen-4-yl)acetamide
5-(3-cyclohexyl-1H-pyrazol-4-yl)-3-(2-methoxyethyl)-1,2,4-oxadiazole
6-methyl-3-[4-(trifluoromethoxy)phenyl]pyridin-2-amine
8-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(dimethylamino)-4-methyl-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}pyrimidine-5-carboxamide
8-[2-(1H-imidazol-1-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-[3,5-bis(trifluoromethyl)phenyl]-5-(piperidine-1-carbonyl)pyrimidin-4-ol
N-[2-methyl-6-(propan-2-yl)phenyl]-2-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}acetamide
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
4-hydroxy-1-(5-phenylpentanoyl)piperidine-4-carboxylic acid
4-(7-fluoro-4-methylquinolin-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(7-methyl-1-benzofuran-2-carbonyl)thiomorpholine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methyl-1H-pyrazole-4-carboxamide
2-(methoxymethyl)-5-{1-[4-(1H-pyrazol-5-yl)phenyl]-1H-imidazol-2-yl}pyrimidine
N,4-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-imidazole-2-carboxamide
2-{[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
2-benzyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-thiazole-4-carboxamide
methyl N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)carbamate
1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-({[1-(2-phenylethyl)piperidin-4-yl]methyl}amino)propan-1-ol
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(1-phenylcyclopropyl)acetamide
5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
ethyl 4-{1-[2-(3,4-dimethylphenyl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
1'-[2-(methylsulfanyl)pyrimidin-4-yl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
4-(2-oxo-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)piperazin-2-one
N,1,3-trimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
methyl 1-({1-[(4-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperidine-4-carboxylate
(1S,5R)-6-(4-methyl-1H-imidazole-2-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[2-(N-methylmethanesulfonamido)ethyl]amino}pyrimidine-5-carboxylic acid
1-cyclopropyl-N-[3-(4-methoxyphenyl)propyl]-5-oxopyrrolidine-3-carboxamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
4-{1-[(2,2-dimethyloxan-4-yl)methyl]azetidin-3-yl}pyridine
3-methoxy-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
2-{4-[(4-cyclopentyl-3-oxopiperazin-1-yl)methyl]phenoxy}propanoic acid
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanoic acid
2-(dimethylamino)-2-(2-fluorophenyl)-N-(3-hydroxypropyl)acetamide
3-hydroxy-3-({[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one