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1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(methanesulfonylmethyl)piperidine
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(1S,5R)-3-(2H-1,3-benzodioxol-5-ylmethyl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-(1H-pyrazol-4-yl)butanamide
dimethyl[1-(1-{[3-(morpholin-4-ylmethyl)phenyl]methyl}piperidin-4-yl)ethyl]amine
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[2-methyl-1-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]methanesulfonamide
2-(propan-2-yl)-8-(quinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-(dimethyl-1,3-oxazole-5-carbonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-(3-methylpyridin-4-yl)piperazine
N-[2-(7-{[4-(dimethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
3-[(2E)-3-phenylprop-2-en-1-yl]-1-(9H-purin-6-yl)piperidine-3-carboxylic acid
3-fluoro-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
(5S,9aS,9bS)-5-[(E)-2-(4-fluorophenyl)ethenyl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-{[(2-fluoroethyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)aniline
1-ethyl-N-[(2-phenoxypyridin-3-yl)methyl]piperidin-4-amine
1-[(2,6-dichloro-3,4-dimethoxyphenyl)methyl]-3-methoxypyrrolidine
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
methyl 3-(4-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
3-(cyclopropylmethyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine-3-carboxylic acid
3-({1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
1-(3,5-dimethylphenyl)-N-(oxan-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(1,3-benzothiazol-2-ylmethyl)(methyl){[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
1-(cyclohexylmethyl)-5-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]piperidin-2-one
N-(3-ethoxy-2-hydroxypropyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
2-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(cyclopropylmethyl)-8-(5-methoxypyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
3,3-diethyl-1-{[(3S,4S)-3-hydroxy-1-[2-oxo-2-(pyrrolidin-1-yl)acetyl]piperidin-4-yl]methyl}urea
1-[(3-chloro-4-methoxyphenyl)methyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
4-({4-methyl-5-[1-(5-propyl-1,2,4-oxadiazol-3-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
(1R,5R)-6-(cyclopropylmethyl)-3-(2-ethylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-1-(4-chloro-2-fluorobenzoyl)-4-cyclopropylpyrrolidin-3-yl]acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]acetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
N-(pyridin-2-ylmethyl)-4-[3-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-cyclopropyl-2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-4-carboxamide
1-methyl-3-[1-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclopentyl-N-[(4,6-dimethylpyridin-3-yl)methyl]-6-oxopiperidine-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[3-(2-methoxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidine-2-carboxamide
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
3-[4-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)piperazine-1-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
6-methyl-2-{2-[2-(quinolin-4-yl)-1H-imidazol-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
ethyl 2-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)amino]acetate
(3S,4S)-4-methyl-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}piperidine-3,4-diol
4-ethyl-5-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3-thiadiazole
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-7-oxo-2-(2-phenoxyacetamido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-2-yl)ethan-1-one