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5-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]isoquinoline
7-oxo-N-(5-oxo-1-propylpyrrolidin-3-yl)-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-ol
(3S,4S)-1-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
5-(4-methylpiperazin-1-yl)-2-[2-(oxolan-3-yl)ethyl]-2,3-dihydropyridazin-3-one
1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]azepan-3-amine
5-(ethylsulfanyl)-N-[2-(4-methylpiperazin-1-yl)ethyl]thiophene-2-carboxamide
N-{1-[1-(but-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
[(3R,5S)-1-[(3-methylquinoxalin-2-yl)methyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
3-methoxy-1-[1-oxo-1-(piperidin-1-yl)propan-2-yl]-1,2-dihydropyridin-2-one
methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](quinoxalin-5-ylmethyl)amine
(3aR,6aR)-2-[1-(4-chlorophenyl)cyclopropanecarbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3S,5S)-1-(propan-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-yl]-1-propylpiperidin-4-amine
methyl 1-[(3S,5S)-1-(3-methylbut-2-en-1-yl)-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-(4-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-4-oxobutyl)-3,4-dihydroquinazolin-4-one
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octane-3-carbonyl]-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
3-(3-fluorophenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
4-[2-(2,2-diphenylethyl)morpholin-4-yl]-6-methylpyrimidin-2-amine
(2S)-2-{[1-(2-aminoethyl)-1H-1,2,3-triazol-4-yl]formamido}-4-methylpentanamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-(2-amino-2-methylpropyl)-2-benzyl-2,8-diazaspiro[5.5]undecan-3-one
(3S,4S)-4-methyl-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidine-3,4-diol
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-(2-methoxyethyl)-4-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[(3S,5S)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
N-[2-(azepan-1-yl)ethyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(propan-2-yl)propanamide
ethyl 3-[(4-fluorophenyl)methyl]-1-[2-(2-oxopiperidin-1-yl)acetyl]piperidine-3-carboxylate
(1-{1-[4-methoxy-3-(morpholin-4-yl)benzoyl]piperidin-4-yl}ethyl)dimethylamine
N-[2-(4-methoxyphenyl)ethyl]-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)acetamide
{2-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-oxoethyl}urea
2-ethyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-5-carboxamide
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
N-[2-hydroxy-2-(3-methoxyphenyl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
(2S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-2-(methoxymethyl)pyrrolidine-1-carboxamide
1-methyl-5-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}piperidin-2-one
2-[3-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenoxy]acetic acid
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-(trifluoromethyl)benzamide
3-tert-butyl-1-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
2-[3-(4-chlorophenyl)-4-methyl-1H-pyrazol-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
3-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1-(thiophen-2-yl)urea
5-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-propylpyrimidin-2-amine
2-(2,8-dimethylquinoline-4-carbonyl)-1,2-oxazolidin-4-ol
3-ethyl-5-methyl-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1,2-oxazole-4-carboxamide
4-(cyclopropylmethyl)-1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
1-[4-(furan-2-yl)phenyl]-N-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-amine