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methyl 2-[1-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-3-oxopiperazin-2-yl]acetate
6-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
N-[1-(3-methylpyridin-2-yl)ethyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
5-{1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-(3-methoxypyrazin-2-yl)-1-[(3-methylphenyl)methyl]piperazin-2-one
1-(propan-2-yl)-4-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-1,4-diazepane
2-(3-methylphenyl)-5-{[4-(oxan-4-yl)piperazin-1-yl]methyl}pyrimidine
[1-(2,3-dihydro-1H-inden-2-yl)-5-[(methylamino)methyl]-1H-1,2,4-triazol-3-yl](phenyl)methanol
1-[1-(2-ethoxyacetyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-(4-{[(adamantan-1-yl)carbamoyl]amino}-3,5-dimethyl-1H-pyrazol-1-yl)acetic acid
6-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
3-benzoyl-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyridine-2-carboxamide
5-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
5-[(3S,4R)-3-carboxy-4-phenylpyrrolidine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylic acid
7-[(4-fluorophenyl)methyl]-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decane
6-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-5,6-dihydro-1,6-naphthyridin-5-one
(3S,4S)-1-(4-cyclopentylpyrimidin-2-yl)-4-(dimethylamino)pyrrolidin-3-ol
(3aR,6aS)-5-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-3-[3-(methylsulfanyl)propanoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(3-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[3-(diethylamino)pyrrolidin-1-yl]-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
1-[2-(1-phenylmethanesulfonylpiperidin-2-yl)ethyl]pyrrolidin-2-one
N,N-dimethyl-3-[methyl(2-phenylethyl)amino]piperidine-1-sulfonamide
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(2-phenylethyl)piperidine-3-carboxamide
1-(1-benzofuran-5-carbonyl)-3-(2-ethylphenoxy)azetidine
ethyl 1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylate
methyl (2S)-1-{2-[4-(4-{[(3S)-2-oxoazepan-3-yl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
6-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyridine-2-carboxylic acid
methyl (2R,4S)-4-hydroxy-1-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidine-2-carboxylate
7-methyl-2-[2-(pyridin-2-yl)piperidine-1-carbonyl]-4H-chromen-4-one
5-ethyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 2-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}amino)benzoate
2-(1,4-dimethylpiperazin-2-yl)-N-[(4-fluorophenyl)methyl]-N-(pyridin-2-ylmethyl)acetamide
1-benzyl-5-(propan-2-yl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(4-fluorophenoxy)-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperidine
4-chloro-3-{[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1-methyl-1H-indazole
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-[2-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}methyl)phenoxy]ethan-1-ol
5-butyl-6-methyl-N4-[3-(morpholin-4-yl)propyl]pyrimidine-2,4-diamine
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
N,N-dimethyl-2-{[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}ethane-1-sulfonamide
1-{2-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
2-cyclobutaneamido-N,N-diethyl-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
N-ethyl-4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxamide
(3aR,6aS)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
methyl 1-methoxy-8-[2-(7-methyl-2-oxo-2H-chromen-4-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(pyridin-2-ylmethyl)acetamide