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2-{[4-(5-acetylthiophene-3-carbonyl)-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide
4-methyl-2-{2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]propanoic acid
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]propanamide
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-phenylpiperidin-4-ol
1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}-3-(3-methoxyphenyl)propan-1-one
3-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-5-methyl-1H-indazole
8-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4-(4-hydroxybenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N-[3-(2-phenylacetamido)phenyl]-1H-1,2,4-triazole-5-carboxamide
3-methyl-4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-3,4-dihydrophthalazine-1-carboxamide
5-(methanesulfonylmethyl)-2-(6-methoxypyridin-3-yl)pyridine
1-(5-chloropyridin-2-yl)-4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperazine
3-[(2R,3R,6R)-5-[(3-fluoro-4-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[2-(2-fluorophenyl)-1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
N-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{1-[4-(3-methylthiophen-2-yl)phenyl]ethyl}morpholine
2-(4-chlorophenyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
2-[2-(2-chloro-3,4-dimethoxyphenyl)-1H-imidazol-1-yl]-N-cyclopropylacetamide
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-(pyridin-3-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-(3-{[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]methyl}phenyl)ethan-1-amine
3-{[(5-tert-butyl-2-hydroxyphenyl)methyl](methyl)amino}-N-methylbutanamide
(4aR,7aS)-4-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(2-chlorophenyl)-5-methyl-4-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1,3-oxazole
[(3R,4S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(2-methylphenyl)methyl]-2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}acetamide
2-(1-{4-[(dipropylamino)methyl]phenyl}-N-methylformamido)-N,2-dimethylpropanamide
(cyclohexylmethyl)(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N,2,5-trimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
1-(3,5-dimethylphenyl)-4-[2-(4-fluorophenyl)-2-hydroxyacetyl]piperazin-2-one
5-{1-[(2-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
5-(2-methylpropyl)-1'-(1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]imidazolidine-2,4-dione
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
2-cyclopropyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
2-(2-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
N-{2-[3-(2-oxopyrrolidin-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
2-[(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
2-(3-hydroxypropyl)-9-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(pyridin-3-yl)-1,3-benzoxazol-5-yl]butan-2-ol
7-(4-methylphenyl)-4-(piperidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
5-(4-fluorophenyl)-N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-(1-ethyl-1H-pyrazol-4-yl)-1-[(2-fluorophenyl)methyl]-1-(2-methoxyethyl)urea
(3aR,6aS)-2-(1-benzofuran-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole