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N-[3-fluoro-5-(trifluoromethyl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
2-[4-(1-cyclopentyl-1H-imidazol-2-yl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
1-(1H-imidazol-2-ylmethyl)-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
4-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
2-[4-(2,6-dimethoxypyrimidine-4-amido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
N-{[3-methyl-7-(1-phenyl-1H-pyrazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide
3-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-N-(1,3-thiazol-2-yl)propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-3-ol
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-cyclohexyl-7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]propanamide
1-[1'-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
methyl 4-(4-{[(2-hydroxyethyl)(thiophen-2-ylmethyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
5-{[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]carbamoyl}thiophene-2-carboxylic acid
3-{5-[(3-methylthiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[2-oxo-6-(pyrrolidin-1-yl)-2,3-dihydro-1H-1,3-benzodiazol-5-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-[3-(1H-imidazol-2-yl)propyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
2-(4-methylpentyl)-4-(thian-4-yl)morpholine
2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine-4-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-(3-phenylpropyl)-4-(pyrimidin-2-yl)morpholine
2-(4-chlorophenoxy)-1-(7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-(4-methanesulfonylphenyl)benzamide
4-[(4-methoxyphenyl)methyl]-1-[(5-methylthiophen-2-yl)methyl]-1,4-diazepan-5-one
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(5-methylpyridin-2-yl)acetamide
(3R,4R)-4-cyclobutyl-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methylpiperidin-4-ol
5-amino-N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-phenyl-1H-pyrazole-3-carboxamide
2-[2-(diethylamino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-propyl-1H-pyrazole-5-carboxamide
1-(4-{4-[(4-hydroxybutyl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
5-ethyl-N4-[2-(pyridin-2-ylsulfanyl)ethyl]pyrimidine-2,4-diamine
2-{4-[2-(benzyloxy)acetyl]morpholin-3-yl}acetic acid
2-(4-fluorophenoxymethyl)-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)piperidine-3-carboxylate
N-(1-benzylpyrrolidin-3-yl)-1-(pyrimidin-2-yl)piperidin-4-amine
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
2-(3-methoxyphenyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
3-(3-fluorophenyl)-N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
3-{2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
3-({[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-1H-1,2,4-triazol-5-amine
N-(1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl)methanesulfonamide
ethyl 3-({1-[(3-fluorophenyl)methyl]-6-oxopiperidin-3-yl}formamido)propanoate
ethyl 4-(oxan-2-ylmethyl)-1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidine-4-carboxylate
2-methyl-4-[4-(oxan-4-yl)piperazin-1-yl]-6-propylpyrimidine
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-1,2,4-triazole
(1S,2R)-2-[methyl({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]cyclohexan-1-ol
5-cyclopropyl-N-(2-hydroxy-2-phenylethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide