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2-cyclopropyl-4-(3-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}piperidin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-(thiophen-3-yl)acetamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-6-(propan-2-yl)-1H-indole-2-carboxamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
5-acetyl-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2,4-dimethyl-1H-pyrrole-3-carboxamide
3-(1H-1,2,4-triazol-3-yl)-N-(2,2,2-trifluoroethyl)benzamide
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[2-(3-hydroxypiperidin-1-yl)-2-oxoethyl]-2,6,6-trimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indol-4-one
5-[2-(3-fluorophenyl)ethyl]-3-(2-methoxyethyl)-1-methyl-1H-1,2,4-triazole
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
N-(2,5-dimethyl-3-{4-phenyl-1-[(2R)-pyrrolidin-2-ylmethyl]-1H-imidazol-5-yl}-1H-pyrrol-1-yl)acetamide
2-butyl-8-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3-(2-oxoazepan-1-yl)propanamide
N-cyclobutyl-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-phenyl-5-[1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrimidin-2-amine
N-(diphenylmethyl)-2-[2-(1H-imidazol-4-yl)acetamido]acetamide
6-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
N-[4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]-2H-1,3-benzodioxole-5-carboxamide
5-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-methylpropanamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-N-(pyridin-2-ylmethyl)cyclopropanamine
1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-{1-[1-(2,2-difluorocyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
3-[3-(pyridin-3-yl)-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[1-({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)pyrrolidin-3-yl]acetamide
methyl 3-(6-methylpyridin-2-yl)benzoate
4-{4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-[(2-fluorophenyl)methyl]acetamide
N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
8-[2-chloro-5-(piperidin-1-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylamino)ethan-1-one
N-(furan-2-ylmethyl)-3-(4-{[(propan-2-yl)carbamoyl]methyl}piperazin-1-yl)propanamide
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-[3-(dimethylamino)pyrrolidin-1-yl]ethan-1-one
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
N-[1-(cyclohex-1-en-1-yl)ethyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylprop-2-en-1-yl)amine
8-(1-benzofuran-5-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-ethyl-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]-1H-pyrazole-4-carboxamide
N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-[(1-benzyl-1H-imidazol-2-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
ethyl 5-(1H-imidazol-2-ylmethyl)-1-[3-(pyridin-3-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[4-(furan-2-carbonyl)piperazin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
4-(1H-imidazol-1-yl)-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]butanamide
dimethyl({4-methyl-5-[1-(thiophene-3-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-[(3R,4S)-4-cyclopropyl-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]-2-ethoxyacetamide
2-cyclopropyl-9-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-{[(6-hydroxynaphthalen-2-yl)methyl](methyl)amino}ethyl)piperidin-2-one
3-methyl-7-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-methyl-9-(4-methyl-1H-imidazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
5-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid