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3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2,6-dimethyl-N-{1-[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}aniline
4-(2-ethoxyphenyl)-5,6-dimethylthieno[2,3-d]pyrimidine
N,2-dimethyl-6-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,6-dihydropyrimidine-5-carboxamide
5-{[2-(2-carboxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}furan-2-carboxylic acid
3-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-(2H-1,3-benzodioxol-5-yl)-5-(but-3-en-1-yl)-3-cyclopropyl-1H-1,2,4-triazole
N-[(2-chlorophenyl)methyl]-1-cyclohexyl-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-({cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-4-methylbenzamide
3-methyl-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
N-benzyl-N,1-dimethyl-5-{methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(azocan-1-yl)-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
[(2-fluoro-4-methoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-ethyl-2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}pyridine-3-carboxamide
6-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
1-{1-[6-(3,4-difluorophenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
4-{[5-(2-methyl-1-benzofuran-5-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
N-cyclopropyl-5-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-indole-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)ethyl]amine
1-ethyl-5-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidine-3-carboxamide
2-{4-[(2,4-difluorophenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
(2S,4S)-4-[4-({[(4-chloro-2-methylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
4-(3-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}propoxy)benzamide
6-fluoro-2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-ethyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-4-ylmethyl)pyridin-2-amine
1-(4-methylphenyl)-4-[2-(2,3,6-trifluorophenyl)acetyl]piperazin-2-one
N-cyclopropyl-5-methyl-N-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}thiophene-2-carboxamide
N4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N2,N2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N,N-dimethylacetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
N-[3-(3,5-dimethylphenoxy)propyl]-N,3-dimethyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-(quinoline-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-fluoro-3-methylphenyl)-6-(1H-pyrazole-4-carbonyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
8-fluoro-N-[2-(furan-2-yl)ethyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
(3S)-1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N,N-dimethylpyrrolidin-3-amine
N-(1,3-benzothiazol-5-yl)-2-(acetamidomethyl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
ethyl 4-{[(1-oxo-1,3-dihydro-2-benzofuran-5-yl)carbamoyl]amino}piperidine-1-carboxylate
N-methyl-3-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
(1S,5R)-6-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
N-{[4-(methylsulfanyl)phenyl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
(1S,6R)-9-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-(1H-pyrrol-2-yl)pyridine-3-carboxamide
1-(3-chloro-2-fluorophenyl)-3-[3-(oxolan-3-yl)propyl]urea
N-[2-(ethanesulfonyl)ethyl]-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(2-{[(2-hydroxyethyl)(propan-2-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol