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butyl 4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxylate
N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-[(1-cyclobutylpiperidin-4-yl)oxy]-4-methoxy-N-(2-methoxyethyl)benzamide
1-{1-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[4-(2,5-dimethylphenyl)piperazin-1-yl]propan-1-one
6-[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
9-methoxy-7-(6-methoxypyridin-2-yl)-4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(8-methoxyquinolin-5-yl)methyl]-N,2-dimethyl-1-benzofuran-5-carboxamide
1-[2-(3-fluorophenyl)ethyl]-5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]piperidin-2-one
4-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}-N-phenylpiperidine-1-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1H-1,2,3-triazole-5-carboxamide
1-{[3-(2,4-dimethoxyphenyl)phenyl]methyl}pyrrolidine
1-[3-(benzyloxy)phenyl]-3-[(1,3-dimethylpyrrolidin-3-yl)methyl]urea
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
7-fluoro-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)quinazolin-4-amine
N-ethyl-1-(1H-indol-2-ylmethyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
6-(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N-methyl-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-[(3-ethoxyphenyl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}pyridine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[3,5-dimethyl-1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]pyridin-3-amine
methyl[(4-methyl-1H-imidazol-5-yl)methyl](quinoxalin-2-ylmethyl)amine
4-{2-[(3-hydroxyphenyl)amino]-6-methylpyrimidin-4-yl}-1,4-oxazepan-6-ol
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
(3aS,6aS)-2-methyl-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-methyl-1H-pyrazol-1-yl)-1-[3-(3-methylphenyl)piperidin-1-yl]propan-1-one
2-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}quinoline
methyl 3-(oxolane-3-amido)-1-(2-phenylethyl)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-chloro-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]thiophene-2-carboxamide
N,2,5,6-tetramethyl-N-[2-(4-methylphenoxy)ethyl]pyrimidin-4-amine
4-(2-methyl-1-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-2-yl)morpholine
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-3-(3-methylpiperidin-1-yl)propanamide
(3R,4S)-4-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1,4-diazepan-1-yl}oxolan-3-ol
3-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-(3-methoxypropyl)-1-[(2-phenylethyl)carbamoyl]piperidine-3-carboxylic acid
N-(1-benzothiophen-2-ylmethyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(1S,5R)-3-(pyridine-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(6-fluoropyridin-3-yl)-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
4-(4-{[(2-methylphenyl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
[5-fluoro-7-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-[(3-methoxyphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)oxane-4-carboxamide
(1R,3S)-3-ethoxy-7-(4-methyl-2-phenylpyrimidine-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
(2S,4S)-4-amino-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
N-(4-{[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}phenyl)acetamide
1-cyclohexyl-1-[2-(ethylsulfanyl)ethyl]-3-(6-methylpyridin-3-yl)urea
N-{1-[7-(1-benzofuran-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}oxolane-3-carboxamide
1-benzyl-N3-ethyl-N5-[(1R)-1-(3-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide