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N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)cyclopropanamine
1-cyclohexyl-4-(pyrimidin-4-yl)piperazin-2-one
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-2-(1-methylpiperidin-4-yl)acetamide
N-{2-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]ethyl}acetamide
(1R,2S,4R)-N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-(2,5-dimethoxyphenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)acetamide
(3R,4R)-1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-4-cyclopropyl-3-methylpiperidin-4-ol
3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(5-methyl-1H-imidazol-4-yl)methyl]acetamide
3-[(2R,3R,6R)-5-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-ethyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1,3-oxazole-4-carboxamide
4-{[5-(1-cyclobutanecarbonylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
4-[2-(furan-2-yl)phenyl]-1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-1,2,3-triazole
6-({[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]amine
(2S,4S)-N-ethyl-4-(4-ethylbenzamido)-1-(furan-3-ylmethyl)pyrrolidine-2-carboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
1-{1-[(3,5-dichloro-2-methoxyphenyl)methyl]pyrrolidin-3-yl}-4-methylpiperazine
2-(2-chlorophenyl)-3-methyl-N-[2-(pyridin-3-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(carbamoylmethyl)-N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3,4-dihydro-2H-1,4-benzoxazine
1-[(4-fluorophenyl)methyl]-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepane
2-amino-6-cyclohexyl-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-cyclopropyl-3-ethoxy-4-(prop-2-en-1-yloxy)-N-(1,3-thiazol-5-ylmethyl)benzamide
1-(6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)butan-1-one
3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
1-[1-(2,2-dimethylbutanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
5-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-phenylpyrimidin-2-amine
3-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-(1,4-dimethylpiperazin-2-yl)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-(2-methylquinolin-5-yl)-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-N,N-dimethylacetamide
1-[(2,6-difluorophenyl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-(2-chloro-4-methylphenyl)-3-(hydroxymethyl)-4-methylpiperazine-1-carboxamide
1-[(3-chloro-5-fluorophenyl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
[2-(1H-imidazol-1-yl)ethyl](methyl){[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
6-{3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-5-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1,3-thiazole
N-cyclopropyl-5-(1H-pyrrole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-(5-fluoro-2-methylphenyl)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(morpholin-4-yl)propanamide
N-[(1-hydroxycyclohexyl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
8-(5-methyl-1,2-oxazole-3-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
(1S,5R)-3-benzyl-6-(morpholine-4-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-5-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-1,3-benzodiazole
3-(2,2-difluoroethyl)-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide